专利号:US-6815214-B2 优先权日:2000-12-29 标 题 :Pharmaceutical uses and synthesis of diketopiperazines 发明人:BOYCE JIM P; HOWBERT J JEFFRY; TABONE JOHN C 权利人:CELLTECH R & D INC 摘要:The synthesis of novel diketopiperazines, their use in inhibiting cellular events such as those involving NFK-α, NFK-β and in the treatment of inflammation events, a combinatorial library of diverse diketopiperazines and process for their synthesis as a library and as individual compounds. In particular novel diketopiperazines are disclosed including their synthesis and use in cellular events such as activation of the transcription factor, nuclear factor, TNF-α, TNF-β and also apoptosis.
专利号:US-7314960-B1 优先权日:2006-09-28 标 题:Catalytic synthesis of oxygenate from alcohol 发明人:LIN SHENG-DIANN; HSIAO TING-CHOU 权利人:UNIV YUAN ZE 摘要:The present invention discloses a method for catalytic synthesis of oxygenate from alcohol. At first, a feeding material comprising at least one alcohol is provided. Next, a copper-containing catalyst is provided and the catalyst further comprises at least one metal element selected from the group consisting of the following: zinc, magnesium, and aluminum elements. Following that, a catalytic reaction of the feeding material over the copper-containing catalyst is carried out to synthesize at least one oxygenate.
专利号:WO-2023099297-A1 优先权日:2021-12-02 标 题:Synthesis of hmo butyrate 发明人:BONRATH WERNER; DE-BOER CASPER; GEBHARD RONALD; GOETZINGER ALISSA; WUESTENBERG BETTINA 权利人:DSM IP ASSETS BV 摘要:The present invention relates to new specific butyrate compounds to a new and improved synthesis of specific butyrates as well their use. Butyrate compounds are very useful compounds.
专利号:US-11370736-B2 优先权日:2019-04-01 标 题:Synthesis of fluoro hemiacetals via transition metal-catalyzed fluoro ester and carboxamide hydrogenation 发明人:DUB PAVEL A; BATRICE RAMI J; GORDON JOHN C 权利人:TRIAD NAT SECURITY LLC 摘要:This application is directed to use of transition metal-ligand complexes to hydrogenate fluorinated esters and carboxamides into fluorinated hemiacetals. Methods for synthesis of certain ligands are also provided.
专利号:US-3887490-A 优先权日:1970-08-27 标 题 :Process for regenerating noble metal catalyst for the synthesis of hydrogen peroxide according to the anthraquinone process 发明人:SCHREYER GERD; THEISSEN FERDINAND; WEIBERG OTTO; WEIGERT WOLFGANG 权利人:DEGUSSA 摘要:In situ regeneration of noble metal catalysts for the synthesis of hydrogen peroxide by the anthraquinone process is provided by employing as the working solution coming from the extraction or desorption step and being introduced into the hydrogenation step a solution which contains at least 250 mg/liter of hydrogen peroxide, to thereby completely regenerate the noble metal catalyst by full capacity of the hydrogenation step.
专利号:WO-2024172286-A1 优先权日:2023-02-14 标题 :Synthesis of photodegradable iron nitrosyl complex and development of pharmaceutical composition for prevention or treatment of vascular diseases, using same 发明人:CHO JAEHEUNG; LEE JUNYEOP; CHOE JISU 权利人:ULSAN NATIONAL INSTITUTE OF SCIENCE AND TECH; ASAN FOUND; UNIV ULSAN FOUND IND COOP 摘要:The present invention relates to a compound represented by chemical formula 1 or a pharmaceutically acceptable salt thereof, a compound represented by chemical Formula 2 or a pharmaceutically acceptable salt thereof, a preparation method thereof, and uses of the compound represented by chemical formula 2 or a pharmaceutically acceptable salt thereof. The compound represented by chemical formula 2 or a pharmaceutically acceptable salt thereof exhibits the effect of releasing nitric oxide in vivo upon light stimulation, thereby dilating blood vessels.
参考标题:A Direct, Versatile, And Chemoselective Synthesis Of Vinylogous Bis- And Monourethanes/amides And β-Keto Esters By Aza-Knoevenagel-Type Reactions Of Tertiary Amides With Enolates 作者:Pei-Qiang Huang,Wei Ou |发布日期:2017.1.18 摘要:Carbanions Generated From Methyl Ketones, Malonic Acid Monoester, 2-Phenylacetate, Or (Benzylsulfonyl)Benzene. Moreover, When Higher Homologous Of Acetate Was Used, Beta-Keto Esters Were Obtained Directly From Amides. The Method Has Been Applied To The One-Step Synthesis Of Several Known Key Intermediates In The Total Synthesis Of Alkaloids And Quinoline Antibiotics. An Efficient And Mild Intramolecular Friedel-Crafts
合成参考文献
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