CAS: 10365-98-7; 3-Methoxyphenylboronic Acid

相似化合物

325142-84-5 438553-44-7 192182-54-0

上下游产品

CAS号2398-37-0 间溴苯甲醚 | CAS号121-43-7 硼酸三甲酯 | CAS号5419-55-6 硼酸三异丙酯 | CAS号325142-84-5 3-甲氧基苯硼酸频哪醇酯 | CAS号100-66-3 苯甲醚 | CAS号73183-34-3 双戊酰二硼 | CAS号13195-76-1 硼酸三异丁酯 | CAS号36282-40-3 3-甲氧苯基溴化镁 | CAS号10540-41-7 4'-Fluoro-3-bip... | CAS号10540-43-9 1-fluoro-4-(3-m... | CAS号1104636-71-6 3-甲氧基苯硼酸甲基亚氨基二乙酸酯 | CAS号459-60-9 4-氟苯甲醚 | CAS号456-49-5 间氟苯甲醚 | CAS号321-28-8 2-氟苯甲醚 | CAS号325142-84-5 3-甲氧基苯硼酸频哪醇酯 | CAS号454-90-0 间三氟甲基苯甲醚 | CAS号38087-96-6 2-联苯-(3-甲氧基)羧酸 | CAS号555-03-3 3-硝基苯甲醚

3-甲氧基苯硼酸频哪醇酯置于polystyrene Boronic Acid,三氟乙酸体系中,用 乙腈 用作溶剂,化学反应 18.0H,以98%的收率获得3-甲氧基苯硼酸
参考文献:Deprotection Of Pinacolyl Boronate Esters By Transesterification With Polystyrene-boronic Acid
标题:Deprotection Of Pinacolyl Boronate Esters By Transesterification With Polystyrene-boronic Acid
摘要:Mild Deprotection Of Pinacolyl Boronate Esters To The Corresponding Boronic Acids Was Achieved In The Presence Of Excess Polystyrene-Boronic Acid Via A Transesterification Process. The Procedure Allows For The Cleavage Of Pinacolyl Boronate Esters In The Presence Of Sensitive Functional Groups. Crown Copyright (C) 2004 Published By Elsevier Ltd. All Rights Reserved.
Doi:10.1016/j.Tetlet.2004.07.014

专利信息

专利号:WO-2025215126-A1
优先权日:2024-04-12
标题:Synthesis of vidofludimus and its calcium salt
发明人：VITT DANIEL; IGLICAR PETRA; GEGE CHRISTIAN; Mühler Andreas; KOHLHOF HELLA; GRÖPPEL MANFRED
权利人:IMMUNIC AG
摘要:The invention relates to the process of preparation of 2-fluoro-4-(3-methoxyphenyl)aniline (3) as an intermediate. Said intermediate 2-fluoro-4-(3-methoxyphenyl)aniline (3) is obtained in a Suzuki coupling reaction from (3-methoxyphenyl)boronic acid (1) and 4-bromo-2-fluoro-aniline (2). The invention further relates to the synthesis of vidofludimus (5) from said intermediate 2-fluoro-4-(3-methoxy-phenyl)aniline (3) and from 1-cyclopentene-1,2-dicarboxylic anhydride (4). The invention further relates to the synthesis of vidofludimus calcium (6) from said vidofludimus (5) and from a calcium salt, preferably Ca(OH)2.

专利号:US-10508092-B2
优先权日:2016-09-02
标题 :Synthesis of novel analogs of diptoindonesin G, compounds formed thereby, and pharmaceutical compositions containing them
发明人：XU WEI; TANG WEIPING; LIU JITIAN; KOLESAR JILL
权利人:WISCONSIN ALUMNI RES FOUND
摘要:Disclosed are unnatural analogs of Diptoindonesin G, methods to make the analogs, pharmaceutical compositions containing the analogs, and methods of using the analogs to inhibit neoplastic cell growth.

专利号:US-11130764-B2
优先权日:2017-02-17
标题 :Analogs of vincamine and uses thereof
发明人：HUIGENS III ROBERT WILLIAM; NORWOOD IV VERRILL M; LUESCH HENDRIK
权利人:UNIV FLORIDA
摘要:The present disclosure provides compounds of any one of Formulae (I′), (I), (IA), (II′), (II), (IIA), (IIIA), (III″), (III′), (III), (IIIA), (IV), (V′), (V), (VI), (VII), (VIII′), (VIII), (IX′), (IX), and (X). The compounds described herein may be useful in treating and/or preventing a broad range of diseases (e.g., proliferative disease (e.g., cancers (e.g., non-small cell lung cancer, or glioma), inflammatory diseases, autoimmune diseases), CNS disorder (e.g., drug addiction), metabolic disorder (e.g., diabetes), or infectious disease (e.g., bacterial infection or parasitic infection (e.g., malaria))). Also provided in the present disclosure are pharmaceutical compositions, methods of synthesis of a compound described herein, kits, methods, and uses including or using a compound described herein.

专利号:US-8030496-B2
优先权日:2005-02-17
标 题:Intermediate compound for synthesis of viridiofungin a derivative
发明人：KATO TATSUYA; KIMURA NOBUAKI; MIZUTANI AKEMI; MAKINO TOSHIHIKO; KAWASAKI KENICHI; FUKUDA HIROSHI; KOMIYAMA SUSUMU; TSUKUDA TAKUO
权利人:CHUGAI PHARMACEUTICAL CO LTD
摘要:A method whereby a compound having HCV replication inhibitory activity and desired optical activity can be synthesized selectively and at high yield in a small number of steps by using a compound having a specific chiral auxiliary as a starting compound is provided. n A compound represented by the formula (1-8): n n n n n n n n n n n n wherein Y represents a group represented by the following formula: n n n n n n n n n n n n n n n n Q represents a protected carbonyl group; D represents —(CH 2 ) m —R′, etc.; and n represents an integer of 0 to 10.

专利号:US-10385087-B1
优先权日:2018-04-26
标题:Xylose derivatives and process for preparation thereof
发明人：HWA KUO-YUAN
权利人:NATIONAL TAIPEI UNIV OF TECHNOLOG; UNIV NAT TAIPEI TECHNOLOGY
摘要:Disclosure of the present invention relates to a method for synthesis of a xylose derivative, which comprises protecting a xylose with a protective group, followed by incorporating to a halogen atom as a leaving group; removing the protective groups and using water-soluble ligands to carry out a Suzuki cross-couplings reaction with a palladium catalyst in a water solution. Ten new xylose derivatives as obtained by the method are also provided.

专利号:US-8207337-B2
优先权日:2007-01-29
标 题:Reagent for organic synthesis reaction containing organic triol borate salt
发明人：MIYAURA NORIO; YAMAMOTO YASUNORI
权利人:MIYAURA NORIO; YAMAMOTO YASUNORI; WAKO PURE CHEM IND LTD
摘要:[Problem] n To provide an organoboron compound-containing reagent for organic synthesis reactions which undergoes no trimerization with dehydration, does not necessitate activation with a base, and is stable and highly active. n [Means for Solving Problems] n The reagent for organic synthesis reactions contains an organic triol borate salt represented by any of the general formulae (I) to (III) and general formula (XVI): (wherein R 1 represents alkyl, alkenyl, etc.; R 2 represents optionally substituted alkyl, alkenyl, alkynyl, etc. or represents hydrogen; m + represents an alkaline metal ion, phosphonium ion, or given ammonium ion; M 2+ represents an alkaline earth metal; X represents halogen or alkoxide; Y represents an alkali metal ion, etc.; A represents optionally substituted methylene; and n represents an integer).