CAS: 4463-42-7; Benzylboronic Acid

上下游产品

CAS号100-44-7 氯化苄 | CAS号121-43-7 硼酸三甲酯 | CAS号6921-34-2 苄基氯化镁 | CAS号1589-82-8 苄基溴化镁 | CAS号6688-98-8 benzyldichloroborane | CAS号351459-60-4 benzylboron dic... | CAS号7732-18-5 水 | CAS号162213-35-6 diisopropyl ben... | CAS号10294-33-4 三溴化硼 | CAS号108-88-3 甲苯 | CAS号87100-28-5 苄基硼酸频哪醇酯 | CAS号22057-44-9 苄基(2-硝基苯基)硫烷 | CAS号2117-39-7 benzyl(chloro)m... | CAS号94242-82-7 2-(1-chloro-2-p... | CAS号7440-22-4 纳米银粉 | CAS号11113-50-1 硼酸 | CAS号134-81-6 联苯甲酰

Benzylboronic Acid Diisopropyl Ester置于硫酸体系中,化学反应生成 苄基硼酸
参考文献:P1 Phenethyl Peptide Boronic Acid Inhibitors Of Hcv Ns3 Protease
标题:P1 Phenethyl Peptide Boronic Acid Inhibitors Of Hcv Ns3 Protease
摘要:A Series Of Peptide Boronic Acids Containing Extended,Hydrophobic P1 Residues Was Prepared To Probe The Shallow,Hydrophobic S1 Region Of Hcv Ns3 Protease. The P-Trifluoromethylphenethyl P1 Substituent Was Identified As Optimal With Respect To Inhibitor Potency For Ns3 And Selectivity Against Elastase And Chymotrypsin. (C) 2002 Published By Elsevier Science Ltd.
DOI:10.1016/s0960-894X(02)00682-0

专利信息

专利号:US-9862745-B2
优先权日:2004-03-30
标题 :Synthesis of boronic ester and acid compounds
发明人：AMMOSCATO VINCE; BISHOP JOHN E; CHIU FANG-TING; GEISER ACHIM; GOMEZ JEAN-MARC; HETT ROBERT; KOELLNER CHRISTOPH; KULKARNI VITHALANAND R; LO YOUNG; MUNK STEPHEN; PICKERSGILL I FRASER
权利人:MILLENNIUM PHARM INC; MILLENNIUM PHARM INC
摘要:The invention relates to the synthesis of boronic ester and acid compounds. More particularly, the invention provides improved synthetic processes for the large-scale production of boronic ester and acid compounds, including the peptide boronic acid proteasome inhibitor bortezomib.

专利号:US-8207337-B2
优先权日:2007-01-29
标 题:Reagent for organic synthesis reaction containing organic triol borate salt
发明人：MIYAURA NORIO; YAMAMOTO YASUNORI
权利人:MIYAURA NORIO; YAMAMOTO YASUNORI; WAKO PURE CHEM IND LTD
摘要:[Problem] n To provide an organoboron compound-containing reagent for organic synthesis reactions which undergoes no trimerization with dehydration, does not necessitate activation with a base, and is stable and highly active. n [Means for Solving Problems] n The reagent for organic synthesis reactions contains an organic triol borate salt represented by any of the general formulae (I) to (III) and general formula (XVI): (wherein R 1 represents alkyl, alkenyl, etc.; R 2 represents optionally substituted alkyl, alkenyl, alkynyl, etc. or represents hydrogen; m + represents an alkaline metal ion, phosphonium ion, or given ammonium ion; M 2+ represents an alkaline earth metal; X represents halogen or alkoxide; Y represents an alkali metal ion, etc.; A represents optionally substituted methylene; and n represents an integer).

专利号:US-2018265546-A1
优先权日:2004-03-30
标题 :Synthesis of boronic ester and acid compounds

专利号:US-2005240047-A1
优先权日:2004-03-30
标 题:Synthesis of boronic ester and acid compounds

专利号:CN-111925385-A
优先权日:2004-03-30
标题 :Synthesis of Boron Ester and Acid Compounds

专利号:US-2020157143-A1
优先权日:2004-03-30
标题 :Synthesis of boronic ester and acid compounds