五氯苯胺置于盐酸,溶剂黄146,Sodium Nitrite体系中,化学反应生成五氯苯硫酚 参考文献:Tadros; Saad,Journal Of The Chemical Society,1954,P. 1155 标题:Tadros; Saad,Journal Of The Chemical Society,1954,P. 1155
专利号:WO-9915510-A1 优先权日:1997-09-24 标 题:Protecting and linking groups for organic synthesis 发明人:TOTH ISTVAN; DEKANY GYULA; KELLAM BARRY 权利人:ALCHEMIA PTY LTD; TOTH ISTVAN; DEKANY GYULA; KELLAM BARRY 摘要:This invention relates to methods for synthesis of organic compounds, and in particular to compounds useful as protecting and linking groups for use in the synthesis of peptides, oligosaccharides, glycopeptides and glycolipids. The invention provides protecting and linking groups which are useful in both solid phase and solution synthesis, and are particularly applicable to combinatorial synthesis. In its most general aspect, the invention provides a cyclic compound of general formula (I).
专利号:US-6765089-B1 优先权日:1997-09-24 标 题 :Protecting and linking groups for organic synthesis on solid supports 发明人:TOTH ISTVAN; DEKANY GYULA; KELLAM BARRY 权利人:ALCHEMIA PTY LTD 摘要:This invention relates to methods for synthesis of organic compounds, and in particular to compounds useful as protecting and linking groups for use in the synthesis of peptides, oligosaccharides, glycopeptides and glycolipids. The invention provides protecting and linking groups that are useful in both solid phase and solution synthesis, and are particularly applicable to combinatorial synthesis.
专利号:WO-2024142008-A1 优先权日:2022-12-29 标 题:A process for the preparation of 2,2' dithiobisbenzanilide 发明人:JAYABALAN LAKSHMANAN; NAMBOODIRI JANARDANAN KAPYUR; CHAUDHURI MONOJIT 权利人:NITREX CHEMICALS INDIA LTD 摘要:The present disclosure relates to a process for the preparation of 2,2'- dithiobisbenzanilide The process involves the hydrolysis of benzothiazole, followed by subsequent oxidation, and the benzoylation of the resulting reaction products to yield 2,2'-dithiobisbenzanilide. The process of the present disclosure is a one-pot synthesis and uses a minimal amount of base for the synthesis of 2,2'-dithiobisbenzanilide. The process is simple, economical, eco-friendly, and commercially scalable.
专利号:WO-9955664-A1 优先权日:1998-04-24 标 题 :Preparation of carbocyclic compounds 发明人:BECKER MARK W; CHAPMAN HARLAN H; KELLY DAPHNE E; KENT KENNETH M; LEW WILLARD; LOUIE MICHAEL S; MCGEE LAWRENCE R; PRISBE ERNEST J; POSTICH MICHAEL J; ROHLOFF JOHN C; SCHULTZE LISA M; YU RICHARD H; ZHANG LIJUN 权利人:GILEAD SCIENCES INC; BECKER MARK W; CHAPMAN HARLAN H; KELLY DAPHNE E; KENT KENNETH M; LEW WILLARD; LOUIE MICHAEL S; MCGEE LAWRENCE R; PRISBE ERNEST J; POSTICH MICHAEL J; ROHLOFF JOHN C; SCHULTZE LISA M; YU RICHARD H; ZHANG LIJUN 摘要:The present invention provides new synthetic methods and compositions. In particular, new methods of preparing intermediates useful in the synthesis of neuraminidase inhibitors and compositions useful as intermediates that are themselves useful in the synthesis of neuraminidase inhibitors are provided.
专利号:US-2024132927-A1 优先权日:2020-12-02 标 题 :Modular glycan production with immobilized bionanocatalysts 发明人:CORGIE STEPHANE CEDRIC; HOEPKER ALEXANDER CHRIS 权利人:ZYMTRONIX CATALYTIC SYSTEMS INC 摘要:The invention provides modular cell-free de-novo synthesis of glycans with immobilized bionanocatalysts. The invention provides materials, and in particular, magnetic materials, for producing glycans of defined length and sequences using one or more enzymes that are immobilized within bionanocatalysts (BNCs) which in turn are embedded within scaffolds to control the synthesis in batch or continuous processes manufacturing. In some embodiments, the scaffolds are high magnetism and high porosity composite blends of thermoplastics or thermosets comprising magnetic particles that form powders. In some embodiments, Selective Laser Sintering (SLS) is used to design and produce objects via 3D printing by sintering composite magnetic powders. The modular flow cells may be mixed and matched for a highly customizable and highly efficient cell-free manufacturing process. In some embodiments the elementary and system modules provided by the invention are employed. In preferred embodiments, human milk oligosaccharides (HMOs) are produced.
专利号:US-7749106-B2 优先权日:2006-03-30 标题 :Molded rubber material for golf ball, method of making the material and golf ball 发明人:SHINDO JUN; NANBA ATSUSHI 权利人:BRIDGESTONE SPORTS CO LTD 摘要:A molded rubber material for a golf ball is obtained by molding and vulcanizing a rubber composition composed of (a) a diene rubber, (b) an α,β-unsaturated carboxylic acid and/or a metal salt thereof, (c) an organic peroxide, and (d) an inorganic oxide. The inorganic oxide is prepared by a plasma process, a laser process or flame synthesis, has an average particle size of at most 200 nm, and is added in an amount of at least 1 wt % based on the zinc acrylate. The molded rubber material has a high hardness, a good resilience, and excellent durability.
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合成参考文献
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