专利号:WO-2017089470-A1 优先权日:2015-11-27 标 题:Process for the synthesis of aryldiazonium salts using nitrogen oxides in oxygen-containing gas streams, especially from industrial waste gases 发明人:HOFMANN DAGMAR; HOFMANN JOSEFA; HEINRICH MARKUS 权利人:Friedrich-Alexander-Universität Erlangen-Nürnberg 摘要:The present invention relates to a process for the synthesis of aryldiazonium salts using nitrogen oxides in oxygen-containing gas streams, especially from industrial waste gases.
专利号:US-2013338369-A1 优先权日:2011-03-07 标 题 :Process for the Synthesis of Aminobiphenylene 发明人:HEINRICH MARKUS; PRATSCH GERALD 权利人:HEINRICH MARKUS; PRATSCH GERALD; BASF SE 摘要:The present invention relates to a process for the synthesis of 2-aminobiphenylene and derivatives thereof by reacting a benzene diazonium salt with an aniline compound under basic reaction conditions.
专利号:WO-2017109658-A1 优先权日:2015-12-23 标 题:Process for the synthesis of patiromer 发明人:GABOARDI MAURO; PRENDIN RICCARDO; CASTALDI MARTA; CASTALDI GRAZIANO 权利人:RJW PHARMA LLC 摘要:The present invention relates to a process for the synthesis of Patiromer, an active ingredient used in the treatment of hyperkalemia in adults.
专利号:WO-2006038872-A1 优先权日:2004-10-08 标 题:New process for the preparation of phosphinic acid 发明人:IOANNIDIS PANAGIOTIS; NILSSON MATHS 权利人:ASTRAZENECA AB; IOANNIDIS PANAGIOTIS; NILSSON MATHS 摘要:A new process for the synthesis of a compound of formula [Chemical formula should be inserted here. Please see paper copy] wherein A represents O or N; R1 represents a C?1#191-C?6#191 alkyl; R2 and R3 each independently represents C?1#191-C?10#191 alkyl, optionally substituted or interrupted by cyclic C?3#191-C?6#191 alkyl, cyclic C?3#191-C?6#191 heteroalkyl, aryl or heteroaryl; and X is selected from F, Cl, Br, or I, by a halogenation procedure comprising the consecutive sequence of following reactions: a) dienalkylation; b) formation of a leaving group on the alcohol function; and c) halogenation, is provided by the present invention as well as the compounds obtainable by the process.
专利号:US-8093421-B2 优先权日:2006-10-27 标题 :Stereoselective one step fluorination process for the preparation of 2-flouropropionate 发明人:LUI NORBERT; PAZENOK SERGII 权利人:LUI NORBERT; PAZENOK SERGII; BAYER CROPSCIENCE AG 摘要:The current invention describes a one-step process for the synthesis of 2-fluoropropionates from lactic acid ester derivatives using TFEDMA.
专利号:US-10611739-B2 优先权日:2016-08-16 标题:Process for preparation of lactone derivatives and intermediates thereof 发明人:CHEN PING; PENG SHAOPING; LI YINQIANG; LI DAFENG; DONG XUEJUN 权利人:PHARMARESOURCES SHANGHAI CO LTD 摘要:A novel process for the preparation of lactone derivatives, and intermediates thereof is described. The lactone derivatives are important precursors for the synthesis of anti-hepatitis C virus agents, including sofosbuvir.
[参考文献]: Junling Li, Et Al. Characterization Of (18)F-Dipicolylamine (Dpa) Derivatives In Cells Infected With Influenza Virus. Nucl Med Biol. 2015 Mar;42(3):283-91.
合成参考文献
摘要:Das, A.; Ramkumar, N.; Veliks, J., Science of Synthesis: Modern Strategies in Organofluorine Chemistry, (2025) 2.