CAS: 207857-15-6; 1,3-Di-Boc-2-(Trifluoromethylsulfonyl)Guanidine

上下游产品

CAS号358-23-6 三氟甲磺酸酐 | CAS号332882-82-3 N,N'-bis(tert-b... | CAS号863891-95-6 N,N-bis(tert-bu... | CAS号219511-71-4 N-B°C-胍 | CAS号24424-99-5 二碳酸二叔丁酯 | CAS号203258-44-0 2-(2-氨基乙基)-1,3-... | CAS号160677-41-8 mono-6-n-dib°C-... | CAS号143824-77-5 N-芴甲氧羰基-N',N''-... | CAS号215050-11-6 1,3-二-B°C-2-(2-羟乙基)胍

Boc-胍置于三氟甲磺酸酐,三乙胺体系中,用 二氯甲烷 用作溶剂,以88%的收率获得1,3-二-Boc-2-(三氟甲基磺酰)胍
参考文献:Guanidinylation Reagents
标题:Guanidinylation Reagents
摘要:三取代n-保护胍和用作胍基化试剂以产生n-保护胍基衍生物的方法.

专利信息

专利号:US-6833445-B2
优先权日:2000-01-21
标题:Guanidinylation, guanidinoglycosides, uses, and methods of assaying their activity
发明人：GOODMAN MURRAY; TOR YITZHAK; BAKER TRACY; LUEDTKE NATHAN
权利人:UNIV CALIFORNIA
摘要:Provided are reagents and methods useful for the synthesis of guanidinylated compounds. Also provided are methods for assaying molecules, including guanidinylated molecules that modulate viral infection and replication.

专利号:US-11999693-B2
优先权日:2015-09-24
标 题:Synthetic sphingolipid-like molecules, drugs, methods of their synthesis and methods of treatment
发明人：EDINGER AIMEE L; HANESSIAN STEPHEN
权利人:UNIV CALIFORNIA; THE UNIV DE MONTREAL
摘要:Small molecules comprised of azacyclic constrained sphingolipid-like compounds and methods of their synthesis are provided. Formulations and medicaments are also provided that are directed to the treatment of disease, such as, for example, neoplasms, cancers, and other diseases. Therapeutics are also provided containing a therapeutically effective dose of one or more small molecule compounds, present either as pharmaceutically effective salt or in pure form, including, but not limited to, formulations for oral, intravenous, or intramuscular administration.

专利号:US-9889182-B2
优先权日:2009-09-15
标 题 :Assisted enzyme replacement therapy
发明人：ESKO JEFFREY D; TOR YITZHAK
权利人:ESKO JEFFREY D; TOR YITZHAK; UNIV CALIFORNIA
摘要:Reagents and methods useful for the synthesis of conjugates comprising guanidinylated cyclic acetals are provided. Also provided are methods for increasing the cellular uptake of various therapeutic compounds and treatment modalities using these conjugates.

专利号:US-8071535-B2
优先权日:2003-09-12
标 题 :Guanidinium derivatives for improved cellular transport
发明人：TOR YITZHAK; LUEDTKE NATHAN
权利人:TOR YITZHAK; LUEDTKE NATHAN; UNIV CALIFORNIA
摘要:Reagents and methods useful for the synthesis of conjugates comprising guanidinylated cyclic acetals are provided. Also provided are methods for increasing the cellular uptake of various therapeutic compounds and treatment modalities using these conjugates.

专利号:FR-2853653-A1
优先权日:2003-04-09
标 题 :CHIRAL DIPHOSPHINES, THEIR PREPARATION AND USES AS LIGANDS IN THE SYNTHESIS OF COMPLEXES FOR ASYMMETRIC CATALYSIS

专利号:FR-2853652-A1
优先权日:2003-04-09
标题:CHIRAL DIPHOSPHINES, THEIR PREPARATION AND USES AS LIGANDS IN THE SYNTHESIS OF COMPLEXES FOR ASYMMETRIC CATALYSIS