CAS: 76497-13-7; Sultamicillin

上下游产品

iodomethyl penicillanate 1,1-dioxide ampicillin sodium salt

Ampicillin Sodium Salt置于n-氯-N-吡啶基乙酰肼,对甲苯磺酸体系中,用 甲醇,N,N-二甲基甲酰胺 作为反应溶剂,化学反应 10.5H,反应生成 舒他西林
参考文献:Synthesis Of 1,1-Dioxopenicillanoyloxymethyl 6-[d-α-(Benzylideneaminophenylacetamido)]Penicillanate And Analogs. New Intermediates In The Preparation Of Sultamicillin
标题:Synthesis Of 1,1-Dioxopenicillanoyloxymethyl 6-[d-α-(Benzylideneaminophenylacetamido)]Penicillanate And Analogs. New Intermediates In The Preparation Of Sultamicillin
摘要:The Synthesis Of Benzylidene Imines Of Sultamicillin And Analogs 1 Is Described. These New Compounds Showed High Stability And Were Prepared Under Very Mild Conditions And High Yields. Furthermore,They Are Convenient Starting Materials For The Preparation Of Sultamicillin 5 (Important Prodrug Of Ampicillin And Sulbactam) As Its Base Form,By Deprotection Of The Amino Group With Girard Reagents. (C) 2001 Elsevier Science Ltd. All Rights Reserved.
DOI:10.1016/s0040-4020(01)00599-3

专利信息

专利号:US-9382288-B2
优先权日:2010-10-06
标题 :Derivatives of steroid benzylamines, having an antiparasitic antibacterial, antimycotic and/or antiviral action
发明人：BECKER KATJA; KRIEG REIMAR; SCHÖNECKER BRUNO
权利人:BECKER KATJA; KRIEG REIMAR; SCHÖNECKER BRUNO; UNIV GIESSEN JUSTUS LIEBIG
摘要:The present invention relates to compounds derived from steroids of the general formula (I) n nwherein L represents a linker and R # represents a steroid residue, the use of compounds of the general formula (I) in medicine and for the prophylaxis and/or the treatment of infectious diseases. Furthermore described are pharmaceutical compositions containing at least one compound of the general formula (I). A further aspect of the invention relates to the synthesis of said compounds of the general formula (I).

专利号:ES-2161602-B1
优先权日:1999-04-08
标 题 :SYNTHESIS OF 6- (D-ALPHA- (BENCILIDENAMINOPHENYLACETAMIDE)) PENICILANATE 1,1-DIOXOPENICILANLANILOXIMETILO AND ANALOGS. NEW INTERMEDIATES FOR SYNTHESIS OF SULTAMICILLIN.

专利号:ES-2161602-A1
优先权日:1999-04-08
标 题 :SYNTHESIS OF 6- (D-ALPHA- (BENCILIDENAMINOPHENYLACETAMIDE)) PENICILINATE 1,1-DIOXOPENICILANLANILOXIMETILO AND ANALOGS. NEW INTERMEDIATES FOR SYNTHESIS OF SULTAMICILLIN.

专利号:JP-2000344783-A
优先权日:1999-04-08
标题:6- [D-α- (benzylideneaminophenylacetamide)] synthesis of 1,1-dioxopenicilanoyloxymethyl penicillate and its analogs, a novel intermediate in the synthesis of sultamicillin

专利号:TR-200000952-A2
优先权日:1999-04-08
标题:Synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (benzylideneamino-phenylacetamido)] penicillanate and the like. New intermediates suitable for the synthesis of sultamicillin.

专利号:TR-200000952-A3
优先权日:1999-04-08
标 题:Synthesis of 1,1-dioxopenicillaniloxymethyl 6- [D-alpha- (benzylideneamino-phenylacetamido)] penicillanate and the like. New intermediates suitable for the synthesis of sultamicillin.