CAS: 133454-47-4; 1-(4-(3-(4-(6-Fluorobenzo[d]Isoxazol-3-yl)Piperidin-1-yl)Propoxy)-3-Methoxyphenyl)Ethan-1-One

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CAS号329977-73-3 3-[1-(3-chlorop... | CAS号498-02-2 香草乙酮 | CAS号84163-13-3 6-氟-3-(4-哌啶基) -... | CAS号109-70-6 1-溴-3-氯丙烷 | CAS号58113-30-7 4-(3-氯丙基氧基)-3-甲氧基苯乙酮 | CAS号1299470-39-5 盐酸伊潘立酮 | CAS号584-08-7 碳酸钾 | CAS号84163-77-9 6-氟-3-(4-哌啶基)-1... | CAS号151719-92-5 3-methoxy-4-(3-... | CAS号534-17-8 碳酸铯 | CAS号133454-55-4 P88 伊潘立酮代谢物

4'-[3-[4-(6-Fluoro-1,2-Benzisoxazol-3-yl)Piperidino]Propoxy]-3'-Methoxyacetophenone Hydrochloride置于三乙胺体系中,用 甲醇 用作溶剂,化学反应生成伊潘立酮
参考文献: An Improved Process For The Preparation Of Iloperidone[fr] Amélioration De Procédé D'élaboration D'Ilopéridone
标题: An Improved Process For The Preparation Of Iloperidone[fr] Amélioration De Procédé D'élaboration D'Ilopéridone
摘要:本发明涉及一种改进的制备公式(i)的依洛噻酮的方法.此外,本发明还提供了一种新型的依洛噻酮盐酸盐多晶形式.

专利信息

专利号:US-9315483-B2
优先权日:2007-09-13
标题 :Synthesis of deuterated catechols and benzo[D][1,3]dioxoles and derivatives thereof
发明人：JONES ANDREW D; ZELLE ROBERT E; SILVERMAN I ROBERT
权利人:CONCERT PHARMACEUTICALS INC
摘要:The present invention provides a convenient and efficient process for the synthesis of d 2 -benzo[d][1,3]dioxoles.

专利号:US-2013261308-A1
优先权日:2012-03-29
标题 :One-pot process for the synthesis of iloperidone
发明人：BETTONI PIERGIORGIO; ROLETTO JACOPO; PAISSONI PAOLO
权利人:PROCOS SPA
摘要:Disclosed is a process for the synthesis of iloperidone starting from 4-hydroxy-3-methoxy acetophenone (acetovanillone), 1-chloro-3-bromo propane and 6-fluoro-3-(4-piperidinyl)-1,2-benzisoxazole hydrochloride, using a one-pot method. n n n n n n n n n n Said process is performed without any intermediate isolation, and is particularly advantageous from the environmental standpoint and in terms of yields, productivity and the purity of the product obtained, both in the reaction mixture and in the crystal isolated.

专利号:US-9884844-B2
优先权日:2012-12-31
标 题:Heterocyclic compounds and methods of use thereof
发明人：FANG QUN KEVIN; CAMPBELL UNA; SPEAR KERRY L
权利人:SUNOVION PHARMACEUTICALS INC; SUNOVION PHARMACEUTICALS INC
摘要:Provided herein are heterocyclyl compounds, methods of their synthesis, pharmaceutical compositions comprising the compounds, and methods of their use. The compounds provided herein are useful for the treatment, prevention, and/or management of various neurological disorders, including but not limited to, psychosis and schizophrenia.

专利号:EP-4630405-A1
优先权日:2022-12-06
标题 :Process for the synthesis of substituted tetrahydrofuran modulators of sodium channels

专利号:WO-2009035652-A1
优先权日:2007-09-13
标 题 :Synthesis of deuterated catechols and benzo[d][1,3] dioxoles and derivatives thereof

专利号:US-5663449-A
优先权日:1989-05-19
标 题 :Intermediate compounds in the synthesis of heteroarylpiperidines, pyrrolidines and piperazines