专利号:US-6525061-B1 优先权日:1999-11-16 标题 :Methods for the solid phase synthesis of 2-amino-4(H)-quinazolinone derivatives 发明人:GOPALSAMY ARIAMALA; YANG HUI Y 权利人:WYETH CORP 摘要:The present invention relates to solid phase synthesis of substituted 2-amino-4(H)-quinazolinone compounds of formula (I):having pharmacological activity, to processes for their preparation, to a combinatorial library and solid phase methods for preparing libraries of the compounds, to utilizing libraries of the compounds for drug discovery, and to pharmaceutical compositions thereof.
专利号:US-6657068-B2 优先权日:2002-03-22 标题:Liquid phase oxidation of halogenated ortho-xylenes 发明人:COLBORN ROBERT EDGAR; HALL DAVID BRUCE; KOCH PETER; OECKEL GERALD 权利人:GEN ELECTRIC 摘要:A method for the manufacture of halophthalic acid by liquid phase oxidation of halo-ortho-xylene is disclosed. The halophthalic acid may be dehydrated to form halophthalic anhydride which is useful in the synthesis of polyetherimide.
专利号:US-6657067-B2 优先权日:2002-03-22 标题 :Method for the manufacture of chlorophthalic anhydride 发明人:COLBORN ROBERT EDGAR; HALL DAVID BRUCE; KOCH PETER; OECKEL GERALD 权利人:GEN ELECTRIC 摘要:A method for the manufacture of chlorophthalic acid by liquid phase oxidation of chloro-ortho-xylene is disclosed. The chlorophthalic acid may be dehydrated to form chlorophthalic anhydride which is useful in the synthesis of polyetherimide.
专利号:US-2002049320-A1 优先权日:2000-04-27 标 题:6-amino-2,4-dioxo-3,4-dihydro-1,3,5-triazine derivatives and methods for the solid phase synthesis thereof 发明人:GOPALSAMY ARIAMALA; YANG HUI Y 权利人:AMERICAN CYANAMID CO 摘要:The present invention relates to substituted 6-amino-2,4-dioxo-3,4-dihydro-1,3,5-triazine compounds of formula (I) n n n having pharmacological activity, to solid phase synthesis methods for their preparation, to combinatorial libraries thereof, utilizing libraries of the compounds for drug discovery, and to pharmaceutical compositions thereof.
专利号:US-7335791-B1 优先权日:2006-11-28 标题 :Process for the synthesis of hydroxy aromatic acids
专利号:US-2008139843-A1 优先权日:2006-11-28 标 题 :Process for the synthesis of hydroxy aromatic acids
参考文献:10.1134/s1070363223040230 摘要:Li J-, Shi Y, Ma L-, Zhou Z-, Ji C. Synthesis, Crystal Structure, and DFT Study of 2-Chloro-N-cyclopropyl-4-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzamide. Russ J Gen Chem. 2023 Apr;93(4):942–8. doi: 10.1134/s1070363223040230.