专利号:US-9328061-B2 优先权日:2012-03-01 标题:Simple organic molecules as catalysts for practical and efficient enantioselective synthesis of amines and alcohols 发明人:HOVEYDA AMIR H; SILVERIO DANIEL L; PILYUGINA TATIANA; TORKER SEBASTIAN; ROBBINS DANIEL 权利人:TRUSTEES BOSTON COLLEGE 摘要:The present invention provides organic molecules and methods thereof for reactions between organoboron reagents and double bonds, such as imines or carbonyls, to stereoselectively provide chiral products including amines and alcohols, entities useful for the preparation of biologically active molecules.
专利号:US-8871966-B2 优先权日:2013-03-15 标 题 :Regiospecific synthesis of terephthalates 发明人:KRAUS GEORGE A; LEE JENNIFER J 权利人:KRAUS GEORGE A; LEE JENNIFER J; UNIV IOWA STATE RES FOUND INC 摘要:A method for preparing 1,4-biscarboxylic acid esters of benzene is provided.
专利号:US-2014275608-A1 优先权日:2013-03-15 标题:Of regiospecific synthesis of terephthalates
专利号:US-5521179-A 优先权日:1991-04-18 标题 :Heterocyclic amides 发明人:BERNSTEIN PETER R; SHAW ANDREW; THOMAS ROYSTON M; WARNER PETER; WOLANIN DONALD J 权利人:ZENECA LTD 摘要:The present invention relates to certain novel heterocyclic amides which are 1-pyridylacetamide compounds of formula I, set out herein, which are inhibitors of human leukocyte elastase (HLE), also known as human neutrophil elastase (HNE), making them useful whenever such inhibition is desired, such as for research tools in pharmacological, diagnostic and related studies and in the treatment of diseases in mammals in which HLE is implicated. The invention also includes intermediates useful in the synthesis of these heterocyclic amides, processes for preparing the heterocyclic amides, pharmaceutical compositions containing such heterocyclic amides and methods for their use.
专利号:US-2015057451-A1 优先权日:2012-03-01 标 题 :Simple organic molecules as catalysts for practical and efficient enantioselective synthesis of amines and alcohols
专利号:WO-2013131043-A1 优先权日:2012-03-01 标 题:Simple organic molecules as catalysts for practical and efficient enantioselective synthesis of amines and alcohols
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