1,3-二溴-2,2-二甲氧基丙烷置于2-[(6-Chloro-2-Phenyl-Quinolin-7-yl)-(3-Chloro-Pyrazin-2-yl)-Methyl]-Isoindole-1,3-Dione体系中,用 Dmf (N,N-Dimethyl-Formamide) 用作溶剂,化学反应 25.0H,反应生成3,3-二甲氧基环丁烷-1,1-二羧酸二异丙酯
参考文献: 6,6-Bicyclic Ring Substituted Heterobicyclic Protein Kinase Inhibitors[fr] Inhibiteurs De La Proteine Kinase Heterobicycliques A Substitution De Noyau Bicyclique 6,6
标题: 6,6-Bicyclic Ring Substituted Heterobicyclic Protein Kinase Inhibitors[fr] Inhibiteurs De La Proteine Kinase Heterobicycliques A Substitution De Noyau Bicyclique 6,6
摘要:该式(I)的化合物及其药用可接受的盐,其中xi,X2,X3,X4,X5,X6,X7,R1和q1在此处定义,抑制igf-1R酶,可用于治疗和/或预防高增殖性疾病,如癌症,炎症,牛皮癣,过敏/哮喘,免疫系统疾病和疾病及中枢神经系统疾病和状况.