CAS: 183208-36-8; 5-Methoxy-7-Azaindole

上下游产品

CAS号124-41-4 甲醇钠 | CAS号183208-35-7 5-溴-7-氮杂吲哚 | CAS号67-56-1 甲醇 | CAS号183208-34-6 5-溴-7-氮杂氧化吲哚 | CAS号183208-32-4 3,3,5-三溴-1H-吡咯[... | CAS号271-63-6 7-氮杂吲哚 | CAS号754214-54-5 5-溴-1-[(1,1-二甲基... | CAS号10592-27-5 2,3-二氢-7-氮杂吲哚 | CAS号183208-38-0 5-甲氧基-1H-吡咯并[2,... | CAS号98549-88-3 5-羟基-7-氮杂吲哚 | CAS号737003-45-1 1-甲基-1H-吡咯并[2,3... | CAS号397842-91-0 5-甲氧基-2-甲基-1H-吡... | CAS号397842-89-6 5-甲氧基-1-(苯磺酰基)-...

7-氮杂吲哚置于palladium 10% On Activated Carbon 吡啶,甲酸,四丁基氟化铵,溴,Sodium,Sodium Hydride,三乙胺,2,3-二氯-5,6-二氰基-1,4-苯醌,Copper(I) Bromide体系中,用 四氢呋喃,二氯甲烷,N,N-二甲基甲酰胺,Mineral Oil 用作溶剂,化学反应 132.0H,反应生成5-甲氧基-7-氮杂吲哚
参考文献:Azaindole Glucokinase Activators
标题:Azaindole Glucokinase Activators
摘要:提供的化合物为公式(I): 以及其中可接受的药用盐,其中取代基如说明书所述.这些化合物以及包含它们的药物组合物,可用于治疗代谢性疾病和障碍,例如,2型糖尿病.

专利信息

专利号:US-2025002518-A1
优先权日:2023-06-16
标 题 :Synthesis of heteroarynes and use thereof
发明人：MATTMILLER ROBERTS COURTNEY COLLEEN; HUMKE JENNA NICOLE; QUINLIVAN ANSEL ANNABEL; BELLI ROMAN GIANCARLO; KARGBO SALLU SO; PLASEK ERIN ELIZABETH
权利人:UNIV MINNESOTA
摘要:Disclosed herein are heterocyclic arynes and methods for preparing the same. Heteroarynes such as 5-membered O- or N-heterocyclic arynes have been considered inaccessible due to ring strain associated with the triple bond. The methods described herein demonstrate that these arynes can be successfully prepared through the utility of pi-backbonding from a transition metal. Synthetic utility of this method has been demonstrated by the facile synthesis and functionalization of heterocycles using these heteroaryne building blocks.

专利号:US-7652137-B2
优先权日:2003-03-06
标 题:Synthesis of 5 substituted 7-azaindoles and 7-azaindolines
发明人：GRACZYK PIOTR PAWEL; KHAN AFZAL; BHATIA GURPREET SINGH
权利人:EISAI R&D MAN CO LTD
摘要:The present invention provides a novel substituted azaindoline intermediate of formula (I) and a method for its synthesis. The novel substitued azaindoline intermediate (I) is provided for use in the manufacture of 5-substituted 7-azaindolines and 5-substituted 7-azaindoles.

专利号:EP-1633750-B1
优先权日:2003-03-06
标题 :Synthesis of 5-substituted 7-azaindoles and 7-azaindolines

专利号:US-12415804-B2
优先权日:2023-06-28
标题 :Compounds for activating a serotonin receptor
发明人：BANISTER SAMUEL; JORGENSEN WILLIAM; TAN JINLONG; WHISH LACHLAN
权利人:Psylo Pty Ltd
摘要:The present disclosure relates generally to compounds, their methods of synthesis, and their use in the treatment of mental illness or central nervous system disorders.

专利号:US-2025163044-A1
优先权日:2021-12-24
标 题:Compounds
发明人：BANISTER SAMUEL; JORGENSEN WILLAM; TAN JINLONG
权利人:Psylo Pty Ltd
摘要:The present disclosure relates generally to compounds, their methods of synthesis, and their use in the treatment of mental illness or central nervous system disorders.

专利号:CN-110128422-B
优先权日:2019-01-04
标题 :Synthesis method of 5-methoxy-7-azaindole