CAS: 406482-19-7; 2-Fluoro-5-Methoxyphenylboronic Acid

上下游产品

1-fluoro-4-methoxybenzene Trimethyl borate (1R,2S)-2-(2-fluoro-5-methoxyphenyl)-1,2-dihydronaphthalen-1-ol 9-(2-fluoro-5-methoxyphenyl)-2-methoxy-7-methylimidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine 2,5-bis(2-fluoro-5-methoxyphenyl)thiophene 2′-amino-6-(2-fluoro-5-methoxyphenyl )-1′,2,2-trimethylspiro[chroman-4,4′-imidazol]-5′(1′H)-one

对氟苯甲醚置于2,2,6,6-四甲基哌啶,正丁基锂,硼酸三异丙酯,盐酸体系中,用 四氢呋喃,正己烷,水 作为反应溶剂,化学反应 2.0H,以65%的收率获得产物2-氟-5-甲氧基苯硼酸
参考文献:General Method For The Synthesis Of Substituted Phenanthridin-6(5H)-Ones Using A Koh-Mediated Anionic Ring Closure As The Key Step
标题:General Method For The Synthesis Of Substituted Phenanthridin-6(5H)-Ones Using A Koh-Mediated Anionic Ring Closure As The Key Step
摘要:Substituted Phenanthridin-6(5H)-Ones Were Obtained In A Two-Step Procedure Involving A Suzuki Cross-Coupling Reaction Followed By A Koh-Mediated Anionic Ring Closure. The Influence Of The Nature And The Position Of The Substituents On The Cyclization Step Were Studied. This Methodology Offers A General And Practical Route To Diversely Substituted Phenanthridin-6(5H)-Ones. (C) 2010 Elsevier Ltd. All Rights Reserved.
DOI:10.1016/j.Tet.2010.05.014

专利信息

专利号:CN-111961073-A
优先权日:2020-09-08
标题 :Continuous synthesis method of arylboronic acid

专利号:CN-111961073-B
优先权日:2020-09-08
标题 :Continuous synthesis method of aryl boronic acid