CAS: 18144-47-3; Tert-Butyl 4-Aminobenzoate

上下游产品

CAS号19756-72-0 4-硝基苯甲酸叔丁酯 | CAS号150-13-0 对氨基苯甲酸 | CAS号59247-47-1 4-溴苯甲酸叔丁酯 | CAS号62-23-7 对硝基苯甲酸 | CAS号1370363-00-0 4-aminobenzoic ... | CAS号75-65-0 叔丁醇 | CAS号122-04-3 对硝基苯甲酰氯 | CAS号16106-38-0 4-氨基苯甲酰氯 | CAS号112888-76-3 4-(2-丙炔氨基)苯甲酸叔丁酯 | CAS号619-45-4 4-氨基苯甲酸甲酯 | CAS号150-13-0 对氨基苯甲酸 | CAS号121506-09-0 tert-butyl 4-(m... | CAS号1141-37-3 Benzoic acid,4-... | CAS号676552-20-8 tert-butyl 4-[2... | CAS号486415-37-6 4-异硫氰基苯甲酸叔丁酯 | CAS号57343-54-1 DQn-1

对氨基苯甲酸置于氯化亚砜,碳酸氢钠体系中,用 二氯甲烷,乙酸乙酯 用作溶剂,化学反应 2.0H,反应生成4-氨基苯甲酸叔丁酯
参考文献:分子内铜介导的碳酰胺羰基化反应制备功能化的吲哚和氮杂吲哚
标题:分子内铜介导的碳酰胺羰基化反应制备功能化的吲哚和氮杂吲哚
摘要:一个主题的不同之处:用于合成功能化的吲哚以及4,5,6和7氮杂吲哚的温和且一般的分子内铜介导的碳镁还原过程是从容易获得的乙酰胺开始的.随后与各种亲电试剂的反应可提供高收率的多官能n杂环.
Doi:10.1002/anie.201304380

专利信息

专利号:US-8809526-B2
优先权日:2010-07-19
标题 :Synthesis of cyclopentaquinazolines
发明人：KERSCHEN JAMES ALAN; BRIDGES ALEXANDER JAMES; DALZIEL SEAN MARK; DAPREMONT Olivier; KIM HYUNJUNG; THOMPSON ANDREW S; ZELLER JAMES ROBERT
权利人:KERSCHEN JAMES ALAN; BRIDGES ALEXANDER JAMES; DALZIEL SEAN MARK; DAPREMONT Olivier; KIM HYUNJUNG; THOMPSON ANDREW S; ZELLER JAMES ROBERT; ONYX PHARMA INC
摘要:A method of producing 6-amino-cyclopenta[g]quinazolines, in enantiomerically enriched form, is provided. In particular, the method may be applicable to the synthesis of N—{N-{4-[N-((6S)-2 -hydroxymethyl-4-oxo-3,4,7,8-tetrahydro-6H-cyclo-penta[g]quinazolin-6-yl)-N-(prop-2 -ynyl)amino]benzoyl}-L-γ-glutamyl}-D-glutamic acid (ONX-0801).

专利号:US-2012196989-A1
优先权日:2005-02-11
标题:Synthesis of homopolymers and block copolymers
发明人：BREITENKAMP KURT; SILL KEVIN N
权利人:BREITENKAMP KURT; SILL KEVIN N; INTEZYNE TECHNOLOGIES INC
摘要:The present invention relates to the field of polymer chemistry and more particularly to homopolymers and block copolymers and methods of preparing the same.

专利号:US-8933227-B2
优先权日:2009-08-14
标题 :Selective synthesis of functionalized pyrimidines
发明人：LINZ GUENTER; KRAEMER GERD; KUSSEROW SABRINA; SCHNAUBELT JUERGEN
权利人:LINZ GUENTER; KRAEMER GERD; KUSSEROW SABRINA; SCHNAUBELT JUERGEN; BOEHRINGER INGELHEIM INT
摘要:The present invention relates to a process for making 2,4-differentiated 5-trifluoromethyl pyrimidines and 2-amino-5-trifluoromethyl-pyrimidine derivatives, which compounds are useful in the preparation of pharmacologically active compounds.

专利号:US-2024059678-A1
优先权日:2021-01-18
标 题 :Synthesis Method for Aminopyrimidine FAK Inhibitor Compound
发明人：DU WU; LV HAIBIN; LI YU; KUANG TONGTAO; GENG XI
权利人:HINOVA PHARMACEUTICALS INC
摘要:A synthesis method for an aminopyrimidine FAK inhibitor compound, relating to the field of pharmaceutical synthesis. In the synthesis method, R1 is hydrogen or a carboxylic acid protecting group, R2 is selected from C1ËœC6 alkyl or C1ËœC6 deuterated alkyl, R3 and R4 are each independently selected from hydrogen or deuterium, and R5 is selected from C1ËœC6 alkyl or C1ËœC6 deuterated alkyl. The synthesis method is simple to operate, and has low costs. The product prepared can obtain a high total yield (≥66%) and a high purity (≥99%), and the product yield and purity are superior to those in the prior art (in the prior art, the total yield is about 11%, and the purity is 99%). The synthesis method achieves excellent effects, can also successfully prepare a final product on kilogram scale, and is suitable for industrial production, having a good application prospect.

专利号:EP-2595966-B1
优先权日:2010-07-19
标题:Synthesis of cyclopentaquinazolines

专利号:US-10308595-B2
优先权日:2013-02-15
标 题:Albicidin derivatives, their use and synthesis
发明人：SUESSMUTH RODERICH; KRETZ JULIAN; SCHUBERT VIVIEN; PESIC ALEXANDER; HUEGELLAND MANUELA; ROYER MONIQUE; COCIANCICH STEPHANE; ROTT PHILIPPE; KERWAT DENNIS; GRAETZ STEFAN
权利人:UNIV BERLIN TECH
摘要:Antibiotically active compounds characterized by general formula (I), wherein X1, BB, BC, BD, BE and X2 are building blocks with D1, D2, D3, D4 or D5 being linkers which include carbon, sulphur, nitrogen, phosphor and/or oxygen atoms and which are covalently connecting the moities BA and BB, BB and BC, BC and BD, BD and BE and BE and BF, respectively, and wherein in particular the building block BC comprises an amino acid derivative. The compounds for use in a method of treatment of diseases, in particular for use in a method of treatment of bacterial infections are also disclosed.