CAS: 4651-81-4; Methyl 2-Aminothiophene-3-Carboxylate

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CAS号40018-26-6 2,5-二羟基-1,4-二噻烷 | CAS号105-34-0 氰乙酸甲酯 | CAS号53982-98-2 methyl 2-cyanob... | CAS号75-07-0 乙醛 | CAS号2125-85-1 1H-吡唑并[3,4-c]吡嗪... | CAS号18740-38-0 2,4-二羟基噻吩[2,3-D]嘧啶 | CAS号18740-39-1 2,4-二氯噻吩[2,3-D]嘧啶 | CAS号81321-10-0 3-异硫氰基噻吩-2-羧酸甲酯 | CAS号126637-07-8 甲基-2-异硫代氰基噻吩-3-羧酸盐 | CAS号14080-50-3 噻吩并[2,3-d]嘧啶-4(3H)-酮 | CAS号55654-21-2 methyl 2-formyl... | CAS号22288-81-9 2-(乙酰氨基)-3-噻吩羧酸甲酯 | CAS号648859-85-2 2-([3-(氯甲基)苯甲酰基... | CAS号845889-21-6 2-[(氨基羰基)氨基]-5-...

Methyl 2-Formylaminothiophene-3-Carboxylate 反应生成 2-氨基噻吩-3-羧酸甲酯
参考文献:Robba M.; Lecomte J. M.; Cugnon De Sevricourt M.,Bull. Soc. Chim. France,1975,No 3-4,Part. 2,587-591
标题:Robba M.; Lecomte J. M.; Cugnon De Sevricourt M.,Bull. Soc. Chim. France,1975,No 3-4,Part. 2,587-591

专利信息

专利号:US-7576211-B2
优先权日:2004-09-30
标题 :Synthesis of thienopyridinone compounds and related intermediates
发明人：DHANOA DALE S; BECKER OREN; NOIMAN SILVIA; CHEN DONGLI; MARANTZ YAEL; SHACHAM SHARON; HEIFETZ ALEXANDER; INBAL BOAZ; BAR-HAIM SHAY; MOHANTY PRADYUMNA; LOBERA MERCEDES; WU LAURENCE
权利人:EPIX DELAWARE INC
摘要:The invention relates to 5-HT receptor agonists and partial agonists. Novel thienopyridinone compounds represented by Formula I, and synthesis and uses thereof for treating diseases mediated directly or indirectly by 5-HT receptors, are disclosed. Such conditions include Alzheimer's disease, cognition disorders, irritable bowel syndrome, nausea, emesis, vomiting, prokinesia, gastroesophageal reflux disease, nonulcer dyspepsia, depression, anxiety, urinary incontinence, migraine, arrhythmia, atrial fibrillation, ischemic stroke, gastritis, gastric emptying disorders, feeding disorders, gastrointestinal disorders, constipation, erectile dysfunction, and respiratory depression. Methods of preparation and novel intermediates and pharmaceutical salts thereof are also included.

专利号:US-2006084805-A1
优先权日:2004-09-30
标题:Synthesis of thienopyridinone compounds and related intermediates

专利号:US-7982040-B2
优先权日:2004-05-17
标题 :Thienopyridinone compounds and methods of treatment
发明人：DHANOA DALE S; BECKER OREN; NOIMAN SILVIA; MOHANTY PRADYUMNA; CHEN DONGLI; LOBERA MERCEDES; WU LAURENCE; MARANTZ YAEL; INBAL BOAZ; HEIFETZ ALEXANDER; BAR-HAIM SHAY; SHACHAM SHARON
权利人:NANOTHERAPEUTICS INC
摘要:The invention relates to 5-HT receptor agonists and partial agonists. Novel thienopyridinone compounds represented by Formula I, and synthesis and uses thereof for treating diseases mediated directly or indirectly by 5-HT receptors, are disclosed. Such conditions include Alzheimer's disease, cognition disorders, irritable bowel syndrome, nausea, emesis, vomiting, prokinesia, gastroesophageal reflux disease, nonulcer dyspepsia, depression, anxiety, urinary incontinence, migraine, arrhythmia, atrial fibrillation, ischemic stroke, gastritis, gastric emptying disorders, feeding disorders, gastrointestinal disorders, constipation, erectile dysfunction, and respiratory depression. Methods of preparation and novel intermediates and pharmaceutical salts thereof are also included.

专利号:WO-2006079916-A1
优先权日:2005-01-26
标 题 :Thieno [2,3-d] pyrimidine compounds as inhibitors of adp-mediated platelets aggregation
发明人：ENNIS MICHAEL DALTON; KORTUM STEVEN WADE; RAHMAN HAYAT; SCHWEITZER BARBARA ANN; TENBRINK RUTH ELIZABETH
权利人:PHARMACIA & UPJOHN CO LLC; ENNIS MICHAEL DALTON; KORTUM STEVEN WADE; RAHMAN HAYAT; SCHWEITZER BARBARA ANN; TENBRINK RUTH ELIZABETH
摘要:Compounds and pharmaceutically acceptable salts of the compounds are disclosed, wherein the compounds have the structure of Formula (I): wherein A1, A2, A3, A4, A5, A6, A7, A8, X4, X6, R2, R4, R5, and R6 are as defined in the detailed description of the invention. Corresponding pharmaceutical compositions, methods of treatment, methods of synthesis, and intermediates are also disclosed.

专利号:US-5179207-A
优先权日:1991-08-19
标 题:Substituted 2-amino-5-maleimido thiophenes and substituted 2-amino-maleimido thiazoles
发明人：KRUTAK JAMES J; WEAVER MAX A
权利人:EASTMAN KODAK CO
摘要:Provided are certain substituted 2-aminothiazoles and 2-aminothiophenes which are useful as red colorants and as intermediates in the synthesis of bathochromic azo dyes. These compounds are prepared by reacting 2-aminothiophenes or 2-aminothiazoles, which contain a primary amino group, with 2-chloro-3-negatively-substituted maleimides. These compounds can be diazotized and coupled with azo components, for example, anilines, 1,2,3,4-tetrahydroquinolines, 2,3-dihydroindoles, and 3,4-dihydro-2H-1,4-benzoxazines to form bathochromic blue-cyan azo dyes.

专利号:US-7407966-B2
优先权日:2004-10-07
标题:Thienopyridinone compounds and methods of treatment
发明人：DHANOA DALE S; BECKER OREN; NOIMAN SILVIA; WU LAURENCE; LOBERA MERCEDES; MOHANTY PRADYUMNA; MARANTZ YAEL; INBAL BOAZ; SHACHAM SHARON; CHEN DONGLI
权利人:EPIX DELAWARE INC
摘要:The invention relates to 5-HT 4 receptor agonists and partial agonists. Thienopyridinone compounds and synthesis and uses thereof for treating diseases mediated directly or indirectly by 5-HT 4 receptors, are disclosed. Such conditions include Alzheimer's disease, cognition disorders, irritable bowel syndrome, Parkinson's disease, nausea, emesis, vomiting, prokinesia, gastroesophageal reflux disease, and nonulcer dyspepsia. Methods of preparation and novel intermediates and pharmaceutical salts thereof are also included.