CAS: 26214-65-3; 3-Furoyl Chloride

相似化合物

498-60-2 488-93-7 636-44-2

上下游产品

CAS号488-93-7 3-糠酸；呋喃-3-甲酸 | CAS号79-37-8 草酰氯 | CAS号4282-28-4 呋喃-2,4-二羧酸 | CAS号4412-91-3 3-呋喃甲醇 | CAS号30614-67-6 3-FURYLMETHYL A... | CAS号142896-19-3 1-(furan-3-yl)-... | CAS号14757-80-3 N,N-dimethylfur... | CAS号148900-66-7 3-Furancarboxam... | CAS号36878-91-8 β-氧代-3-呋喃丙酸乙酯 | CAS号39244-10-5 3-(3-呋喃基)丙烯酸 | CAS号498-60-2 3-糠醛 | CAS号614-98-2 3-呋喃羧酸乙酯 | CAS号14313-09-8 1-呋喃-3-乙酮

3-糠酸置于氯化亚砜,N,N-二甲基甲酰胺体系中,用 二氯甲烷 用作溶剂,化学反应 16.0H,反应生成3-呋喃甲酰氯
参考文献:降压的1-酰基-4-[2-(1,4-苯并二恶烷-2-基)-2-羟乙基氨基]-哌啶.
标题:降压的1-酰基-4-[2-(1,4-苯并二恶烷-2-基)-2-羟乙基氨基]-哌啶.
摘要:制备了几种1-酰基-4-[2-(1,4-苯并二恶烷-2-基)-2-羟基-乙基氨基]哌啶,并且许多化合物在自发性高血压大鼠(shr)中显示出降压活性.该活性对(2S,2R)对映异构体是特异性的.关于所选化合物的一般药理评估和配体结合数据表明,α1和β拮抗活性的程度适中.α1拮抗作用可能不足以解释shr中的降血压活性.
Doi:10.1002/jps.2600760110

专利信息

专利号:US-9765027-B2
优先权日:2014-08-22
标题 :Substituted 1-arylethyl-4-acylaminopiperidine derivatives as opioid/alpha-adrenoreceptor modulators and method of their preparation
发明人：VARDANYAN RUBEN S; HRUBY VICTOR J
权利人:THE ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIV OF ARIZAONA; UNIV ARIZONA
摘要:The invention provides compounds that bind with high affinities to the μ-, δ- and κ-opioid receptors and α 2 -adrenoreceptor. In addition to providing these compounds with novel pharmacological binding properties, the invention also describes detailed novel methods for the preparation of representative compounds and a scheme for the synthesis of related compounds that bind to the opioid receptors and/or α 2 -adrenoreceptor.

专利号:US-2004254162-A1
优先权日:2001-07-16
标 题 :Oxazolidinone derivatives as antimicrobials
发明人：MEHTA ANITA; ARORA SUDERSHAN R; DAS BISJAWIT; RAY ABHIJIT; RUDRA SONALI; RATTAN ASHOK
摘要:The present invention relates to certain substituted phenyl oxazolidinones and to processes for the synthesis of the same. This invention also relates to pharma-ceutical compositions containing the compounds of the present invention as anti-microbials. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms such as Bacterioides spp. and Clostridia spp. species, and acid fast organisms such as Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.

专利号:US-6956040-B2
优先权日:2001-07-16
标题:Oxazolidinone piperazinyl derivatives as potential antimicrobials
发明人：MEHTA ANITA; ARORA SUDERSHAN K; DAS BISWAJIT; RAY ABHIJIT; RUDRA SONALI; RATTAN ASHOK
权利人:RANBAXY LAB LTD
摘要:The present invention relates to certain substituted phenyl piperazinyl oxazolidinones, for example, to those having the structure of Formula I n n nwith the variables as defined within, and to processes for the synthesis of the same. This invention also relates to pharmaceutical compositions containing the compounds of the present invention as antimicrobials. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms such as Bacterioides spp. and Clostridia spp. species, and acid fast organisms such as Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.

专利号:US-6734307-B2
优先权日:2000-07-17
标 题:Oxazolidinone derivatives as antimicrobials
发明人：MEHTA ANITA; SUDERSHAN ARORA K; DAS BISWAJIT; RAY ABHIJIT; RUDRA SONALI; RATTAN ASHOK
权利人:RANBAXY LAB LTD
摘要:The present invention relates to certain substituted phenyl oxazolidinones and to processes for the synthesis of the same. This invention also relates to pharmaceutical compositions containing the compounds of the present invention as antimicrobials. The compounds are useful antimicrobial agents, effective against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci, streptococci and enterococci as well as anaerobic organisms such as Bacterioides spp. and Clostridia spp. species, and acid fast organisms such as Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium spp.

专利号:WO-2012009519-A1
优先权日:2010-07-15
标题:Synthesis and anticancer activity of aryl and heteroaryl-quinolin derivatives

专利号:CN-103347859-B
优先权日:2010-07-15
标 题:Synthesis and Anticancer Activity of Aryl and Heteroaryl Quinoline Derivatives