CAS: 19881-18-6; 1-Isothiocyanato-4-(4-Nitrophenoxy)Benzene

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CAS号62939-03-1 3-[[4-(4-nitrop...

4-硝基-4'-氨基二苯醚置于吡啶体系中,用 5,5-Dimethyl-1,3-Cyclohexadiene,水 用作溶剂,化学反应 2.75H,反应生成硝硫氰醚
参考文献:新的4 [4-(4-硝基苯氧基)苯基]-5-取代的-2 H-1,2,4-三唑-3-硫酮的合成及其驱虫药的评价
标题:新的4 [4-(4-硝基苯氧基)苯基]-5-取代的-2 H-1,2,4-三唑-3-硫酮的合成及其驱虫药的评价
摘要:合成了新颖的4-[4-(4-硝基苯氧基)苯基]-5-取代的-2 H-1,2,4-三唑-3-硫酮在5-位含有不同取代基的文库 .进行机械化学处理以合成目标化合物 8(ap),并通过研磨法和常规方法比较了产率.通过单晶x射线研究分析了中间体异硫氰酸根合-4-(4-硝基苯氧基)苯 6 的结构 .通过光谱和元素分析表征标题化合物,并进一步评估其作为体外驱虫药的功效.化合物 8C,8J,8K,8L 和 8M 表现出明显的驱虫活性.
Doi:10.1007/s11164-015-2123-1

专利信息

专利号:US-2008176865-A1
优先权日:2005-06-15
标 题:Substituted arylpyrazoles
发明人：BILLEN DENIS; BOYLE JESSICA; CRITCHER DOUGLAS JAMES; GETHIN DAVID MORRIS; HALL KIM THOMAS; KYNE GRAHAM MICHAEL
权利人:PFIZER LTD
摘要:This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which the cyclopropyl ring is substituted at the angular position, and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.

专利号:US-7645786-B2
优先权日:2005-06-15
标题:Substituted arylpyrazoles
发明人：BILLEN DENIS; BOYLE JESSICA; CRITCHER DOUGLAS JAMES; GETHIN DAVID MORRIS; HALL KIM THOMAS; KYNE GRAHAM MICHAEL
权利人:PFIZER
摘要:This invention relates to a range of 1-aryl-4-cyclopropylpyrazoles in which the cyclopropyl ring is substituted at the angular position, and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes to their synthesis and their use as parasiticides.

专利号:CN-1191541-A
优先权日:1995-06-14
标题 :Synthesis modification of spinosyn compounds