CAS: 52-52-8; 1-Aminocyclopentanecarboxylic Acid

相似化合物

117322-30-2 35264-09-6 17191-44-5

上下游产品

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在 水,Potassium Hydroxide体系中,用 四氢呋喃 作为反应溶剂,化学反应 6.0H,以0.77 G的收率获得产物环亮氨酸
参考文献:环烷烃螺乙内酰脲和哌啶基螺乙内酰脲的微波辅助合成作为限制性α-氨基酸的前体
标题:环烷烃螺乙内酰脲和哌啶基螺乙内酰脲的微波辅助合成作为限制性α-氨基酸的前体
摘要:在微波辅助条件下,由环烷酮 9 和哌啶酮 10 合成环烷烃螺乙内酰脲 3 和哌啶螺乙内酰脲 4.结果与在热条件下获得的结果进行比较.环烷螺乙内酰脲 3 用 Boc 基团进行 N-保护并在碱性条件下水解,以非常好的总产率 (76-94%) 获得五,六和七元环限制性 α-氨基酸 12.
DOI:10.3998/ark.5550190.0012.221

专利信息

专利号:US-12351573-B2
优先权日:2019-05-09
标 题:Compounds for use in synthesis of peptidomimetics
发明人：AL-ABED YOUSEF; CHENG KAI FAN
权利人:FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH
摘要:Synthesis of O-benzotriazole and O-imidazole synthons are described. Uses of synthons in synthesis of azapeptides and other peptidomimetics, azapeptides and other peptidomimetics synthesized from the synthons and uses of azapeptides and other peptidomimetics are also described.

专利号:US-2023159450-A1
优先权日:2020-05-08
标 题 :Dimers for use in synthesis of peptidomimetics
发明人：AL-ABED YOUSEF; ALTITI AHMAD
权利人:FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH
摘要:Dimers for use in synthesis of peptidomimetics are described. Uses of dimers as synthons in synthesis of azapeptides and other peptidomimetics, azapeptides and other peptidomimetics synthesized from the dimers and uses of azapeptides and other peptidomimetics are also described.

专利号:WO-2008138621-A3
优先权日:2007-05-16
标题 :Synthesis of aminocyclopentane carboxylic acids
发明人：SCHANN STEPHAN; MAYER STANISLAS; ROOME STEPHEN
权利人:FAUST PHARMACEUTICALS; SCHANN STEPHAN; MAYER STANISLAS; ROOME STEPHEN
摘要:The invention relates to efficient methods of synthesis for compounds which are effectors of central nervous system receptors sensitive to neuroexcitatory amino acids such as glutamate or for synthetic precursors or intermediates of these compounds. In particular, the invention provides synthetic strategies and methods which can suitably be applied in the stereoselective synthesis of compounds included in the chemical family of aminocyclopentane tricarboxylic acids.

专利号:US-5880295-A
优先权日:1994-02-16
标 题 :Process for the preparation of diamine intermediates useful in the synthesis of HIV protease inhibitors
发明人：KALTENBACH III ROBERT FRANK
权利人:DU PONT PHARM CO
摘要:The present invention provides a process for the preparation of compounds of formula (V) below, and analogs thereof, which are useful as intermediates for the synthesis of HIV protease inhibitors, including cyclic ureas. ##STR1##

专利号:US-9475837-B2
优先权日:2011-12-23
标题 :Process for the synthesis of therapeutic peptides
发明人：HURLEY FIONN; WEGNER KATARZYNA; FOLEY PATRICK
权利人:IPSEN MFG IRELAND LTD
摘要:The present invention relates to a process for the large-scale synthesis of therapeutic peptides using a Sieber Amide resin, which comprises solid-phase Fmoc-chemistry.

专利号:US-9174943-B2
优先权日:2010-02-24
标 题 :Processes for the synthesis of diarylthiohydantoin and diarylhydantoin compounds
发明人：JAIN RAJENDRA PARASMAL; ANGELAUD REMY; THOMPSON ANDREW; LAMBERSON CAROL; GREENFIELD SCOTT
权利人:JAIN RAJENDRA PARASMAL; ANGELAUD REMY; THOMPSON ANDREW; LAMBERSON CAROL; GREENFIELD SCOTT; MEDIVATION PROSTATE THERAPEUTICS INC
摘要:Processes are provided for the synthesis of diarylthiohydantoin and diarylhydantoin compounds. Medicinal products containing the same find particular use in treating prostate cancer, including castration-resistant prostate cancer and/or hormone-sensitive prostate cancer.