专利号:US-11542283-B2 优先权日:2018-05-28 标题 :Synthesis of peptide borate ester compound and use thereof 发明人:QIN YANRU 权利人:JIANGSU CHIA TAI FENGHAI PHARMACEUTICAL CO LTD 摘要:Provided are a peptide borate ester compound or a pharmaceutically acceptable salt thereof, a preparation method therefor, and pharmaceutical use thereof. The peptide borate ester compound or pharmaceutically acceptable salt thereof has a structure as shown in Formula (I), and is useful in the preparation of proteasome inhibitors to treat solid tumors and hematoma.
专利号:US-7122694-B2 优先权日:1998-11-06 标 题 :Hydroboronation process 发明人:MARCUCCIO SEBASTIAN MARIO; RODOPOULOS MARY; WEIGOLD HELMUT 权利人:BORON MOLECULAR PTY LTD 摘要:The invention relates to processes for the synthesis of aryl or alkene borates which comprises reacting: (i) an olefinic compound having a halogen or halogen-like substituent in a vinylic substitution position, or (ii) an aromatic ring having a halogen or halogen-like substituent in a ring substitution position, with a disubstituted monohydroborane in the presence of a Group 8-11 metal catalyst. The invention also relates to the use of these borates in coupling reactions. The invention further relates to certain disubstituted monohydroboranes and aryl or alkene borates.
专利号:US-2021214377-A1 优先权日:2018-05-28 标题 :Synthesis of peptide borate ester compound and use thereof
专利号:CA-3101824-A1 优先权日:2018-05-28 标题 :Synthesis of peptide borate ester compound and use thereof
专利号:WO-2019228299-A1 优先权日:2018-05-28 标 题:Synthesis and uses of peptide borate ester compound
专利号:CN-115785137-A 优先权日:2018-05-28 标 题:Synthesis and application of a kind of peptide boronate compound
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