专利号:US-6521664-B1 优先权日:1999-12-08 标 题:Pesticidal activity of functionalized alkenes 发明人:LINDERMAN RUSSELL J 权利人:UNIV NORTH CAROLINA STATE 摘要:The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as “pesticidal compoundsâ€?). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
专利号:US-11542279-B2 优先权日:2016-06-06 标 题:Solid forms of ceftolozane and processes for preparing 发明人:MALONEY KEVIN MATTHEW; SIROTA ERIC M; VARSOLONA RICHARD J; GAUTHIER JR DONALD R; REN HONG 权利人:MERCK SHARP & DOHME; MERCK SHARP & DOHME LLC 摘要:The instant invention is related to a novel solid form of ceftolozane sulfate (the DMAc solvate of ceftolozane sulfate (Form 3)), compositions comprising ceftolozane sulfate DMAc solvate (Form 3), synthesis of Form 3 and an improved crystallization process using Form 3 to prepare ceftolozane sulfate Form 2. Novel compositions also include ceftolozane sulfate solid Form 3 and/or other crystalline and amorphous solid forms of ceftolozane.
专利号:WO-2025056767-A1 优先权日:2023-09-15 标题 :Process for the preparation of enantiomerically enriched aliphatic amines 发明人:BOU HAMDAN FARHAN; GODINEAU EDOUARD; SMEJKAL TOMAS; DUMEUNIER RAPHAEL; BOUSSEMGHOUNE MOHAMED ABDELOUAHAB; BLUM MATHIAS 权利人:SYNGENTA CROP PROTECTION AG 摘要:The present invention relates to a process for the preparation of enantiomerically enriched cyclobutylamines of formula (I) from α-tertiary cyclobutanones and reacting said enantiomerically enriched cyclobutylamines to enantiomerically enriched cyclobutylamides. Such compounds are useful intermediates in the synthesis of microbiocidal thiazole compounds.
专利号:US-6660770-B2 优先权日:1999-12-08 标题:Pesticidal activity of functionalized alkenes 发明人:LINDERMAN RUSSELL J; ROE R MICHAEL; THOMPSON DEBORAH M; VANDERHEREHEN MATTHEW 权利人:UNIV NORTH CAROLINA STATE 摘要:The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as “pesticidal compoundsâ€?). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
专利号:US-2022372509-A1 优先权日:2019-08-23 标题:Brown marmorated and harlequin stink bug pheromone enzyme synthesis and uses thereof 发明人:THOLL DOROTHEA; LANCASTER JASON 权利人:VIRGINIA POLYTECHNIC INSTITUTE AND STATE UNIV 摘要:Described herein are engineered polynucleotides and vectors capable of encoding one or more engineered harlequin and/or brown marmorated stink bug pheromone synthesis enzymes. Also described herein are engineered harlequin and/or brown marmorated stink bug pheromone synthesis enzymes. Also described herein are methods of making modified plants capable of expressing one or more harlequin and/or brown marmorated stink bug pheromone synthesis enzymes.
专利号:US-10906880-B2 优先权日:2016-01-26 标题:Kind of isothiazole oxime ether-containing strobilurin derivatives and its preparation methods and application 发明人:FAN ZHIJIN; CHEN LAI; GUO XIAOFENG; ZHU YUJIE; QIAN XIAOLIN; MA LIUYONG; ZHANG NAILOU; WANG HAIXIA; ZHANG ZHIMING; XU JINGHUA; SONG YINQI 权利人:UNIV NANKAI 摘要:The present invention is that provided a synthesis method of a series of isothiazole oxime ether containing strobilurin derivatives IV. The present invention relates to 3,4-dichloroisothiazolyl oxime ether strobilurin derivatives, and their chemical structural formula is as shown by IV. n n n n n n n n n n The invention discloses the structural formula of the above compound, the synthesis method and the use as an insecticide, a fungicide, an anti-plant virus agent, and an agriculturally acceptable auxiliary or synergist and a commercial insecticide. The use of a fungicide, an anti-plant virus agent and an acaricide in combination for controlling agricultural, forestry, horticultural plant pests, diseases, virus diseases and preparation methods.
1: Christian S, Pradhan P, Jans U. Investigation of the Nucleophilic Attack of Dichlorvos by Reduced Sulfur Species using (1)H NMR. J Agric Food Chem. 2017 Dec 9. doi: 10.1021/acs.jafc.7b04749. [Epub ahead of print] doi: 10.18295/squmj.2017.17.03.006. Epub 2017 Oct 10. 4: Kanu KC, Ijioma SN, Atiata O. Haematological, Biochemical and Antioxidant Changes in Wistar Rats Exposed to Dichlorvos Based Insecticide Formulation Used in Southeast Nigeria. Toxics. 2016 Nov 29;4(4). pii: E28. doi: 10.3390/toxics4040028. 5: Akande MG, Ahmed US. Taurine abated subacute dichlorvos toxicity. Toxicol Rep. 2017 Aug 30;4:463-466. doi: 10.1016/j.toxrep.2017.08.001. eCollection 2017.
合成参考文献
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