CAS: 366-99-4; 3-Fluoro-4-Methoxyaniline

上下游产品

2-氟-4-硝基苯甲醚 2-Fluoro-1-Methoxy-4-Nitrobenzene 455-93-6
2-氟苯甲醚 1-Fluoro-2-Methoxybenzene 321-28-8
N-(3-氟-4-甲氧基苯基)乙酰胺 N-(3-Fluoro-4-Methoxyphenyl)Acetamide 452-15-3
2,4-二氟苯甲醚 2,4-Difluoroanisole 452-10-8
甲氧苯胺 4-Methoxy-Aniline 104-94-9

3-氟-4-甲氧基苯乙酮置于sodium Tetrahydroborate,O-新戊酰羟铵三氟甲磺酸盐,水体系中,化学反应 8.0H,反应生成3-氟-4-甲氧基苯胺
参考文献:使用氧化还原活性胺化试剂进行选择性碳-碳键胺化:苯胺的直接方法†
标题:使用氧化还原活性胺化试剂进行选择性碳-碳键胺化:苯胺的直接方法†
摘要:胺是化学合成中最基本的基序之一,通过选择性 C-C 键裂解引入胺结构单元可以通过直接骨架修饰从简单的碳氢化合物中构建含氮化合物.在此,我们报告了一种使用氧化还原活性胺化试剂通过施密特型重排从烷基芳烃制备苯胺的新方法,该试剂很容易从羟胺中制备.在温和条件下,由相应的烷基芳烃或苯甲醇制备伯胺和仲胺.也展示了改造的非常好兼容性和有价值的应用.
Doi:10.1002/cjoc.202100430

专利信息

专利号:US-2005234244-A1
优先权日:2004-04-20
标题:Synthesis of COX-2 and FAAH inhibitors
发明人：BARTOLINI WILMIN; CALI BRIAN M; CHEN BARBARA; CHIEN YUEH-TYNG; CURRIE MARK G; MILNE G T; PEARSON JAMES P; TALLEY JOHN J; ZIMMERMAN CRAIG
权利人:BARTOLINI WILMIN; CALI BRIAN M; CHEN BARBARA; CHIEN YUEH-TYNG; CURRIE MARK G; MILNE G T; PEARSON JAMES P; TALLEY JOHN J; ZIMMERMAN CRAIG
摘要:Methods for preparing indoles that are useful COX-2 inhibitors and intermediates useful in such methods are described.

专利号:US-2005026965-A1
优先权日:2000-12-29
标 题 :Pharmaceutical uses and synthesis of nicotinanilide-N-oxides

专利号:US-2023104311-A1
优先权日:2020-02-17
标题:Novel 6-substituted 7-deazapurines and corresponding nucleosides as medicaments
发明人：HERDEWIJN PIET; GROAZ ELISABETTA; QINGFENG LI
权利人:UNIV LEUVEN KATH
摘要:The present invention relates to the synthesis of 6-substituted 7-deazapurines and their corresponding nucleosides by coupling aryl or alkyl Grignard reagents with halogenated purine nucleosides in the presence of iron or an iron/copper mixture such as Fe(acac)3/CuI. The present invention also relates to pharmaceutical compositions comprising said compounds and the use of said pharmaceutical compositions to treat or prevent viral infections.

专利号:US-2003004189-A1
优先权日:2000-12-29
标 题 :Pharmaceutical uses and synthesis of nicotinanilide-N-oxides

专利号:WO-2006050120-A2
优先权日:2004-11-01
标题:Synthesis of cox-2 and faah inhibitors

专利号:US-2010063105-A1
优先权日:2000-12-29
标题 :Pharmaceutical uses and synthesis of nicotinanilide-n-oxides