CAS: 4441-56-9; Cyclohexylboronic Acid

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87100-15-0 446065-11-8 122035-40-9

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CAS号22092-92-8 N,N-二异丙基氨基硼烷 | CAS号7732-18-5 水 | CAS号931-50-0 环己基溴化镁 | CAS号931-51-1 环己基氯化镁 | CAS号110-83-8 环己烯 | CAS号36140-19-9 氯代二环己基硼烷 溶液 | CAS号7727-37-9 氮气 | CAS号19573-22-9 Cyclohexane, azido | CAS号68498-84-0 boric acid-carbon | CAS号446065-11-8 环己基三氟硼酸钾 | CAS号446065-11-8 环己基三氟硼酸钾 | CAS号75-46-7 三氟甲烷 | CAS号401-75-2 (三氟甲基)环己烷 | CAS号30169-75-6 环己基硼酸-1,3-丙二醇酯 | CAS号87100-15-0 环己烷硼酸频那醇酯 | CAS号5458-48-0 4-环己基-1-硝基苯 | CAS号3116-98-1 2-cyclohexylcyc... | CAS号18594-05-3 4'-环己基苯乙酮 | CAS号20681-51-0 3-环己基丙酸甲酯 | CAS号1759-68-8 N-环己基苯甲酰胺

三环己基硼烷置于水,碘体系中,化学反应生成 环己基硼酸
参考文献:Metallorganische Derivate Des Acetylens. Iv. ber Einige AlkylBor-Acetylene
标题:Metallorganische Derivate Des Acetylens. Iv. ber Einige AlkylBor-Acetylene
摘要:Abstractdie Darstellung Und Die Eigenschaften Von Bis‐(Dialkylbor)‐acetylenen Werden Beschrieben. Eine Reihe Von Dialkylborjodiden Und Dialkylborsäuren Wird Erstmalig Dargestellt Und Charakterisiert. Die Eigenschaften Der Dargestellten Verbindungen Sind Typisch Für Gemischte Organische Borine,Deren Herausragende Eigenschaft Die Neigung Zur Bildung Gleichartig Substituierter Borine Ist.
DOI:10.1002/zaac.19592990310

专利信息

专利号:US-9862745-B2
优先权日:2004-03-30
标题 :Synthesis of boronic ester and acid compounds
发明人：AMMOSCATO VINCE; BISHOP JOHN E; CHIU FANG-TING; GEISER ACHIM; GOMEZ JEAN-MARC; HETT ROBERT; KOELLNER CHRISTOPH; KULKARNI VITHALANAND R; LO YOUNG; MUNK STEPHEN; PICKERSGILL I FRASER
权利人:MILLENNIUM PHARM INC; MILLENNIUM PHARM INC
摘要:The invention relates to the synthesis of boronic ester and acid compounds. More particularly, the invention provides improved synthetic processes for the large-scale production of boronic ester and acid compounds, including the peptide boronic acid proteasome inhibitor bortezomib.

专利号:WO-2022170218-A1
优先权日:2021-02-05
标题:Intramolecular cyclization for general synthesis of bicyclic alkyl bioisostere boronates
发明人：QIN TIAN; YANG YANGYANG; TSIEN JET
权利人:UNIV TEXAS
摘要:Disclosed herein are methods of synthesizing compounds of the formula (I) wherein the variables are defined herein. Also provided are compounds produced using these methods. In some aspects, the methods provided herein may be used to install aryl bioisosteres.

专利号:US-9243004-B2
优先权日:2011-07-22
标题 :Synthesis of boronic esters and boronic acids using grignard reagents
发明人：CLARY JACOB W; SINGARAM BAKTHAN
权利人:CLARY JACOB W; SINGARAM BAKTHAN; UNIV CALIFORNIA
摘要:Boronic esters and boronic acids are synthesized at ambient temperature in an ethereal solvent by the reaction of Grignard reagents with a boron-containing substrate. The boron-containing substrate may be a boronic ester such as pinacolborane, neopentylglycolborane, or a dialkylaminoborane compound such as diisopropylaminoborane. The Grignard reagents may be pre-formed or generated from an alkyl, alkenyl, aryl, arylalkyl, heteroaryl, vinyl, or allyl halide compound and Mg 0 . When the boron-containing substrate is a boronic ester, the reactions generally proceed at room temperature without added base in about 1 to 3 hours to form a boronic ester compound. When the boron-containing substrate is a dialkylaminoborane compound, the reactions generally proceed to completion at 0° C. in about 1 hour to form a boronic acid compound.

专利号:US-8207337-B2
优先权日:2007-01-29
标 题:Reagent for organic synthesis reaction containing organic triol borate salt
发明人：MIYAURA NORIO; YAMAMOTO YASUNORI
权利人:MIYAURA NORIO; YAMAMOTO YASUNORI; WAKO PURE CHEM IND LTD
摘要:[Problem] n To provide an organoboron compound-containing reagent for organic synthesis reactions which undergoes no trimerization with dehydration, does not necessitate activation with a base, and is stable and highly active. n [Means for Solving Problems] n The reagent for organic synthesis reactions contains an organic triol borate salt represented by any of the general formulae (I) to (III) and general formula (XVI): (wherein R 1 represents alkyl, alkenyl, etc.; R 2 represents optionally substituted alkyl, alkenyl, alkynyl, etc. or represents hydrogen; m + represents an alkaline metal ion, phosphonium ion, or given ammonium ion; M 2+ represents an alkaline earth metal; X represents halogen or alkoxide; Y represents an alkali metal ion, etc.; A represents optionally substituted methylene; and n represents an integer).

专利号:US-2018265546-A1
优先权日:2004-03-30
标题 :Synthesis of boronic ester and acid compounds

专利号:US-2005240047-A1
优先权日:2004-03-30
标 题:Synthesis of boronic ester and acid compounds