专利号:DD-294717-A5 优先权日:1990-05-28 标 题 :PROCESS FOR SYNTHESIS OF SUBSTITUTED PYRAZOLE-4-CARBONSAEUREAL CYLINDERS
专利号:US-7427625-B2 优先权日:2006-02-08 标 题 :Substituted thiatriazaacenaphthylene-6-carbonitrile kinase inhibitors 发明人:CONNOLLY PETER J; EMANUEL STUART L; HAYDEN STUART; JOHNSON SIGMOND G; LAGU BHARAT; MIDDLETON STEVEN A; PANDEY NIRANJAN B; POWELL MARK T 权利人:JANSSEN PHARMACEUTICA NV 摘要:The present invention is directed to substituted thiatriazaacenaphthylene-6-carbonitrile compounds of formula (I): n nand forms thereof, their synthesis and use for treating, preventing or ameliorating a chronic or acute protein kinase mediated disease, disorder or condition.
专利号:US-7803832-B2 优先权日:2004-03-18 标题 :N-(1-arylpyrazol-4L)sulfonamides and their use as parasiticides 发明人:CRITCHER DOUGLAS JAMES; WALSHE NIGEL DEREK ARTHUR; LAURET CHRISTELLE 权利人:PFIZER; PFIZER PROD INC 摘要:The invention relates to a sulfonamide compound of formula (I) or a pharmaceutically, veterinarily or agriculturally acceptable salt or solvate thereof, where the groups R 1 -R 5 are described in the description, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides.
参考标题:Metal-Free Synthesis Of Biaryl- And Teraryl-Cored Diarylmethanes By Ring Transformation Of 2H-Pyran-2-Ones 作者:Fateh Singh,Priyanka Kole |发布日期:2019.3 摘要:Efficient Metal-Free Approach For The Synthesis Of Functionalized Biaryl-Cored Diarylmethanes Is Described By The Ring Transformation Of 2H-Pyran-2-Ones Using 4-Phenylbutan-2-One As Carbanion Source. Moreover, 2H-Pyran-2-Ones Were Reacted With 1,3-Diphenylacetone In The Presence Of Base To Achieve Functionalized Teraryl-Cored Diarylmethanes. All The Ring Transformation Reactions Were Performed Under Mild
合成参考文献
摘要:Singh, F. V., Science of Synthesis Knowledge Updates, (2021) 1, 154. 摘要:von Angerer, S., Science of Synthesis Knowledge Updates, (2011) 1, 156.