专利号:US-3755368-A 优先权日:1971-03-01 标题:Formylation of carboxylic compounds with carbon monoxide 发明人:HUBER J 权利人:PENICK S & CO 摘要:A METHOD FOR THE PREPARATION OF 2-FORMYL ESTERS. THE METHOD INVOLVES THE REACTION OF A CARBOXYLIC COMPOUND HAVING AT LEAST TWO HYDROGEN ATOMS ON THE CARBON ATOM ALPHA TO THE CARBOXYL GROUP WITH CARBON MONOXIDE, PREFERABLY UNDER PRESSURE. THE METHOD IS PARTICULARLY APPLICABLE TO THE PREPARATION OF 2-FORMYL-4-ETHYLENEDIOXY VELERATES. THESE COMPOUNDS ARE USEFUL AS INTERMEDIATES IN THE SYNTHESIS OF VALUABLE INSECTICIDES, E.G., 5-BENZYL-3FURYLMETHYL CHRYSANTHEMATE.
专利号:US-5637757-A 优先权日:1995-04-11 标 题 :One-pot synthesis of ring-brominated benzoate compounds 发明人:HILL JOHN E; FAVSTRITSKY NICOLAI A; MAMUZIC RASTKO I; BHATTACHARYA BHABATOSH 权利人:GREAT LAKES CHEMICAL CORP 摘要:A method of preparing tetrabromobenzoate compounds from tetrabromophthalic anhydride by reacting tetrabromophthalic anhydride with alcohol in the presence of a decarboxylation catalyst. The reaction may be carried out in an excess of alcohol, or with a near stoichiometric amount of alcohol by performing the reaction in an inert solvent.
专利号:US-2004053999-A1 优先权日:1997-09-17 标题 :Novel compounds and methods for synthesis and therapy 发明人:BISCHOFBERGER NORBERT W; DAHL TERRENCE C; HITCHCOCK MICHAEL J M; KIM CHOUNG U; LEW WILLARD; LIU HONGTAO; MILLS ROGER G; WILLIAMS MATTHEW A 摘要:Novel compounds are described. The compounds generally comprise an acidic group, a basic group, a substituted amino or N-acyl and a group having an optionally hydroxylated alkane moiety. Pharmaceutical compositions comprising the inhibitors of the invention are also described. Methods of inhibiting neuraminidase in samples suspected of containing neuraminidase are also described. Antigenic materials, polymers, antibodies, conjugates of the compounds of the invention with labels, and assay methods for detecting neuraminidase activity are also described.
专利号:US-6225341-B1 优先权日:1995-02-27 标 题:Compounds and methods for synthesis and therapy 发明人:BISCHOFBERGER NORBERT W; KIM CHOUNG U; LEW WILLARD; LIU HONGTAO; WILLIAMS MATTHEW A 权利人:GILEAD SCIENCES INC 摘要:Novel compounds are described. The compounds generally comprise an acidic group, a basic group, a substituted amino or N-acyl and a group having an optionally hydroxylated alkane moiety. Pharmaceutical compositions comprising the inhibitors of the invention are also described. Methods of inhibiting neuraminidase in samples suspected of containing neuraminidase are also described. Antigenic materials, polymers, antibodies, conjugates of the compounds of the invention with labels, and assay methods for detecting neuraminidase activity are also described.
专利号:WO-9632368-A1 优先权日:1995-04-11 标题:One-pot synthesis of ring-brominated benzoate compounds
专利号:US-4093622-A 优先权日:1975-05-19 标题 :Pyridine esters of cyclopropane-carboxylic acid 发明人:HENRICK CLIVE A; STAAL GERARDUS B 权利人:ZOECON CORP 摘要:Heterocyclic organic esters and thioesters characterized by the presence of one or two cyclopropane moieties, synthesis thereof, and compositions thereof for the control of mites and ticks.
[参考文献]: Hajime Maeda, Et Al. Hydrogen-Bonding Directed, Regioselective Photocycloaddition Reactions Of Cyanonaphthalenes With Furanmethanols. Photochem Photobiol Sci. 2011 Sep;10(9):1445-9. [参考文献]: Ivan Salmerón, Et Al. Sensory Characteristics And Volatile Composition Of A Cereal Beverage Fermented With Bifidobacterium Breve Ncimb 702257. Food Sci Technol Int. 2014 Apr;20(3):205-13. [参考文献]: Jai K Chavda, Et Al. Synthetic Studies Towards The Core Structure Of Nakadomarin A By A Thioamide-Based Strategy. European J Org Chem. 2014 Jan;2014(1):129-139.
合成参考文献
摘要:Parmeggiani, F.; Galman, J. L.; Montgomery, S. L.; Turner, N. J., Science of Synthesis, (2019) , 397. 摘要:Kwiecień, H. U., Science of Synthesis: Knowledge Updates, (2024) 3, 175.