CAS: 19044-88-3; Oryzalin

上下游产品

4,N4-di-n-propylsulfonyl chloride3,5-dinitro-N4,N4-di-n-propylsulfonyl chloride potassium 4-chloro-3,5-dinitrobenzene sulfonate di-n-propylamine 4-chloro-3,5-dinitrobenzenesulfonic acid4,N4-di-n-propylsulfonyl chloride3,5-dinitro-N4,N4-di-n-propylsulfonyl chloride

Potassium 4-Chloro-3,5-Dinitrobenzenesulfonate置于五氯化磷,氨体系中,用 甲醇,二氯甲烷 用作溶剂,化学反应 8.0H,反应生成氨磺乐灵
参考文献:Synthesis And Antitubulin Activity Of N-And N4-Substituted 3,5-Dinitro Sulfanilamides Against African Trypanosomes And Leishmania
标题:Synthesis And Antitubulin Activity Of N-And N4-Substituted 3,5-Dinitro Sulfanilamides Against African Trypanosomes And Leishmania
摘要:Thirty Analogues Of N-1-Phenyl-3,5-Dinitro-N-4,N-4-Di-N-Propylsulfanilamide (Gb-Ii-5,Compound 3),A New Antikinetoplastid Antimitotic Agent,Have Been Synthesized And Evaluated. The Addition Of Simple Functional Groups To The N1 Aromatic Ring Generally Decreases Antiparasitic And Antimitotic Potency,But Placement Of A Dibutyl Substituent At The N4 Nitrogen To Give N-1-Phenyl-3,5-Dinitro-N-4,N-4-Di-N-Butylsulfanilamide (Compound 35) Augments Antitrypanosomal And Antileishmanial Activity. Compound 35 Possesses Ic50 Values Of 0.12 And 2.6 Mum Against Cultured T. Brucei And L. Donovani Amastigote-Like Forms,Surpassing The Activity Of Compound 3 Against These Parasites By 3.4-And 1.9-Fold,Respectively. Compound 35 Inhibits The Assembly Of Leishmanial Tubulin With An Ic50 Of 6.9 Mum And Displays Antimitotic Effects In Cultured T Brucei As Assessed By Flow Cytometry,But Shows Little Effect On Purified Mammalian Tubulin,And Displays 100-Fold Selectivity For Trypanosomes Over Two Mammalian Cell Lines. Although 3 And 35 Were Not Effective In Initial In Vivo Antitrypanosomal Assays,The In Vitro Potency And ;Selectivity Of These Compounds Make N-1-Aryl-3,5-Dinitro-N-4,N-4-Dialkylsulfanilamides A Promising New Class Of Antikinetoplastid Agents That Act On Parasite Tubulin.
Doi:10.1021/jm0304461

专利信息

专利号:US-2015245570-A1
优先权日:2012-11-15
标题:Reverse synthesis of breeding lines
发明人：VOGELAAR ARIE; VERHOEF RUDOLF; SCHUT JOHANNES WILHELMUS; DIRKS ROBERT HÉLÈNE GHISLAIN
权利人:RIJK ZWAAN ZAADTEELT EN ZAADHANDEL BV
摘要:The invention relates to a method for producing parental lines for a hybrid organism. This method is based on the segregation of individual alleles in the spores produced by a desired plant and/or in the progeny derived from the self-pollination of that desired plant, and on the subsequent identification of suitable progeny plants in one generation, or in a limited number of inbred cycles. The invention further relates to a method for reconstructing a partially heterozygous starting organism.

专利号:WO-2024256370-A1
优先权日:2023-06-13
标 题 :Synthesis of glufosinate using an amidase-based process
发明人：ZIMMERMANN GUNTHER; POTT MORITZ STEFAN
权利人:BASF SE
摘要:The present invention relates to a method of preparing glufosinate, comprising the steps of hydrolysing an N-carbamoyl glufosinate amide with an Amidase enzyme to form an N- carbamoyl amino acid compound followed by cleaving off the carbamoyl moiety of said N- carbamoyl amino acid compound.

专利号:US-2025120400-A1
优先权日:2021-12-10
标题:Synthesis of glufosinate using a hydantoinase-based process
发明人：DITRICH KLAUS; BREUER MICHAEL; POTT MORITZ STEFAN; ZIMMERMANN GUNTHER; SEEMAYER STEFAN
权利人:BASF SE
摘要:The present invention relates to a method of manufacturing glufosinate, comprising the steps of hydrolysing a hydantoin with a Hydantoinase enzyme to form a N-carbamoyl amino acid compound followed by cleaving off the carbamoyl moiety of said N-carbamoyl amino acid compound.

专利号:US-11919928-B2
优先权日:2016-03-16
标题 :Method for producing dihydrotentoxin
发明人：KUBO TAKASHI; MACHIDA MASAYUKI; FUJIOKA TOMONORI; YAMAGUCHI Shigenari; KAWAI KIYOSHI
权利人:KUMIAI CHEMICAL INDUSTRY CO
摘要:An object of the present invention is to identify an enzyme having activity of synthesizing dihydrotentoxin that is a tentoxin precursor and an enzyme having activity of synthesizing tentoxin using dihydrotentoxin as a substrate. The present invention concerns a tentoxin synthesis-related gene encoding a protein comprising the amino acid sequence of SEQ ID NO: 16 and having activity of nonribosomal peptide synthesis of dihydrotentoxin and a tentoxin synthesis-related gene encoding a protein comprising the amino acid sequence of SEQ ID NO: 18 and having activity of converting dihydrotentoxin to tentoxin.

专利号:US-2021386068-A1
优先权日:2018-11-07
标题 :Compositions comprising pyridine carboxylate herbicides and very long chain fatty acid (vlcfa) synthesis inhibitor herbicides
发明人：KISTER JEREMY; SATCHIVI NORBERT M
权利人:CORTEVA AGRISCIENCE LLC
摘要:Disclosed herein are compositions comprising (a) a pyridine carboxylate herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof and (b) a VLCFA synthesis inhibitor herbicide. Also disclosed herein are methods of controlling undesirable vegetation, comprising applying to vegetation or an area adjacent the vegetation or applying in soil or water to control the emergence or growth of vegetation (a) a pyridine carboxylate herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof, and (b) a VLCFA synthesis inhibitor herbicide.

专利号:US-2021352899-A1
优先权日:2018-11-07
标题 :Compositions comprising pyridine carboxylate herbicides and fatty acid and lipid synthesis inhibitor herbicides
发明人：KISTER JEREMY; SATCHIVI NORBERT M
权利人:CORTEVA AGRISCIENCE LLC
摘要:Disclosed herein are compositions comprising (a) a pyridine carboxylate herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof and (b) a fatty acid and lipid synthesis inhibitor (FA/LSI) herbicide, an agriculturally acceptable salt or ester thereof, or mixtures thereof. Also disclosed herein are methods of controlling undesirable vegetation, comprising applying to vegetation or an area adjacent the vegetation or applying in soil or water to control the emergence or growth of vegetation (a) a pyridine carboxylate herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof and (b) a fatty acid and lipid synthesis inhibitor (FA/LSI) herbicide, an agriculturally acceptable salt or ester thereof, or mixtures thereof.