专利号:WO-0009116-A1 优先权日:1998-08-14 标 题:Grp receptor ligands 发明人:XIANG JIA-NING; KARPINSKI JOSEPH M; CHRISTENSEN SIEGFRIED B IV 权利人:SMITHKLINE BEECHAM CORP; XIANG JIA NING; KARPINSKI JOSEPH M; CHRISTENSEN SIEGFRIED B IV 摘要:Novel GRP receptor antagonists are provided. Methods of using the present compounds to antagonize GRP receptors are also provided. The present invention further involves the synthesis of the present compounds.
专利号:US-12227528-B2 优先权日:2017-11-09 标 题:Glucose-sensitive albumin-binding derivatives 发明人:KRUSE THOMAS; KOFOD-HANSEN MIKAEL; MUENZEL MARTIN WERNER BORCHSENIUS; THOEGERSEN HENNING; SAUERBERG PER; EWALD JAKOB; BEHRENS CARSTEN; HOEG-JENSEN THOMAS; BALSANEK VOJTECH; DROBNAKOVA ZUZANA; DROZ LADISLAV; HAVRANEK MIROSLAV; KOTEK VLADISLAV; STENGL MILAN; SNAJDR IVAN; DRUSANOVA HANA 权利人:NOVO NORDISK AS 摘要:This invention relates to glucose-sensitive albumin-binding diboron conjugates. More particularly the invention provides novel diboron compounds, and in particular diboronate or diboroxole compounds, useful as intermediate compounds for the synthesis of diboron conjugates.
专利号:KR-102325534-B1 优先权日:2019-10-11 标题 :Synthesis of Sulfones and Sulfonyl Derivatives using Sodium (tert-butyldimethylsilyl)oxymethanesulfinate
专利号:US-8399680-B2 优先权日:2007-09-28 标 题:Arylamine synthesis method 发明人:TAILLEFER MARC; XIA NING 权利人:TAILLEFER MARC; XIA NING; CENTRE NAT RECH SCIENT 摘要:The invention relates to a method for preparing arylamines and, in particular, a method for preparing aniline and anilines substituted on the aromatic ring from ammonia, under easily-industrialized mild conditions with good selectivity and yields, in the presence of a catalytic system including a copper complex.
专利号:CN-108129478-B 优先权日:2018-01-12 标题:A kind of copper process for catalytic synthesis of organic sulphones and application
专利号:CN-109232343-A 优先权日:2018-10-24 标 题 :A method for copper-catalyzed synthesis of aromatic/alkane 2,2,2-trifluoroethyl selenide and its application in pesticides
参考标题:Copper(II)-Catalyzed Single-Step Synthesis Of Aryl Thiols From Aryl Halides And 1,2-Ethanedithiol 作者:Yajun Liu,Jihye Kim,Heesun Seo,Sunghyouk Park,Junghyun Chae |发布日期:2015.7.6 摘要:Single‐step Synthesis Of Aryl Thiols From Aryl Halides Has Been Developed Employing Copper(II) Catalyst And 1,2‐ethanedithiol. The Key Features Are Use Of Readily Available Reagents, A Simple Operation, And Relatively Mild Reaction Conditions. This New Protocol Shows A Broad Substrate Scope With Excellent Functional Group Compatibility. A Variety Of Aryl Thiols Are Directly Prepared From Aryl Halides In High
合成参考文献
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