专利号:US-6946562-B2 优先权日:2001-12-12 标 题:Synthesis of peptoid substituted azole compounds 发明人:DIEHL DONALD R; NIGER ROBERT J; SCHMITTHENNER HANS F; SONNEFELD WILLIAM J; DUNLAP RICHARD P 权利人:EASTMAN KODAK CO 摘要:Disclosed is a process for the preparation of a peptoid substituted azole compound comprising reacting an amino functionalized azole compound with a resin bound peptoid oligomer bearing a terminal halogen substituent followed by cleavage of the resultant product from the resin surface using a fluorinated organic acid in an inert solvent.
专利号:US-2003187188-A1 优先权日:2001-12-12 标 题:Synthesis of peptoid substituted azole compounds
专利号:US-5928851-A 优先权日:1996-06-20 标题:Photographic couplers which release useful groups anchiomerically and their synthesis 发明人:ALLWAY PHILIP ARTHUR 权利人:EASTMAN KODAK CO 摘要:The present invention describes an image dye-forming coupler of formula (I) wherein L is an oxymethylene or oxycarbonyl group; n is 0 or 1; COUP is a coupler moiety and R1 and R2 are the same or different and are groups selected such that (a) together with the nitrogen atom a good leaving group is formed; (b) at least one of them contains a PUG linked to an electrophilic center (E); and (c) neither R1 nor R2 is a hydrogen atom wherein the coupler is a DIAR coupler from which inhibitor is released from a coupling-off group after a timed delay which results from an additional reaction step. Such delay permits control over the time of release, rate of release and rate of diffusion of a photographically useful group (PUG) without altering the nature of the PUG itself. A method of preparing the coupler is also described wherein the two parts of the molecule can be built up separately and combined in a single reaction allowing ready access to a large variety of possible structures.
专利号:EP-1319975-A1 优先权日:2001-12-12 标 题 :Synthesis of peptoid substituted azole compounds
专利号:US-6190852-B1 优先权日:1999-12-28 标 题:Photographic element containing nitrogen heterocycle substituted cyan coupler and process 发明人:MURA ALBERT J; SCARINGE RAYMOND P; HARDER JOHN W 权利人:EASTMAN KODAK CO 摘要:Disclosed is a photographic element comprising a light-sensitive silver halide emulsion layer having associated therewith a cyan dye-forming coupler represented by Formula (I): n wherein: n each R 1 and R 3 is an independently selected substituent, m is 0 to 5, and p is 0 to 2; n X is hydrogen or a coupling-off group; n W and W 2 represent the atoms necessary to complete rings; and n R 2 is an alkyl or aryl group. n The element provides desirable hue properties and ease of synthesis.
摘要:Marks - Marks JG, DeLeo VA. Contact and Occupational Dermatology, 2nd Ed. St. Louis: Mosby, 1997. 摘要:Gigiena i Sanitariya. For English translation, see HYSAAV., 51(9)(71), 1986 摘要:National Technical Information Service., OTS0570977