CAS: 272-49-1; 4-Azaindole

相似化合物

1018950-15-6 4943-67-3 73177-35-2

上下游产品

CAS号123846-65-1 2-(3-硝基吡啶-2-基)乙腈 | CAS号849353-49-7 (2-trimethylsil... | CAS号65156-92-5 N,N-dimethyl-2-... | CAS号112671-57-5 (2-Trimethylsil... | CAS号1219095-87-0 N-B°C-2-甲基-3-氨基吡啶 | CAS号68-12-2 N,N-二甲基甲酰胺 | CAS号150281-83-7 3-硝基-2-乙烯基吡啶 | CAS号5470-18-8 2-氯-3-硝基吡啶 | CAS号24509-73-7 1-乙酰基-1H-吡咯并[3,... | CAS号18699-87-1 2-甲基-3-硝基吡啶 | CAS号55052-27-2 6-氯-1H-吡咯并[2,3-B]吡啶 | CAS号55052-24-9 7-氮杂吲哚-7-氧化物 | CAS号143468-10-4 methyl 6-iodopy... | CAS号192189-15-4 3-溴-1H-吡咯并[3,2-... | CAS号23612-34-2 N,N-dimethyl-1-... | CAS号23688-47-3 3-溴-4-氮杂吲哚 | CAS号824-51-1 6-甲基-7-氮杂-吲哚 | CAS号276862-85-2 4-氮杂吲哚-3-甲醛 | CAS号1000340-28-2 3-溴-6-甲基-7-氮杂吲哚 | CAS号1116136-36-7 4-氮杂吲哚-4-氧化物

2-溴-3-氨基吡啶置于copper(L) Iodide,四(三苯基膦)钯,Potassium Tert-Butylate,三乙胺体系中,用 四氢呋喃,乙腈 用作溶剂,化学反应 8.0H,反应生成4-氮杂吲哚
参考文献:Compounds For Using In Imaging And Particularly For The Diagnosis Of Neurodegenerative Diseases
标题:Compounds For Using In Imaging And Particularly For The Diagnosis Of Neurodegenerative Diseases
摘要:该发明涉及公式(II)的化合物,用于影像学,特别是用于诊断神经退行性疾病.

专利信息

专利号:US-11427596-B2
优先权日:2019-07-19
标 题:Metal-free solvent-free synthesis of fused-pyrido heterocycles and biomedical applications
发明人：CHELVAM VENKATESH; DUDHE PREMANSH; KRISHNAN MENA ASHA; SONAWANE AVINASH
权利人:INDIAN INSTITUTE OF TECH INDORE
摘要:Embodiments herein provide fused-pyrido heterocycles such as azaindoles, carboline derivatives, furo[b]pyridines or furo[b]pyridine-isatin hybrids of Formula I.Embodiments also relate to a process for a synthesis of variety of complex pyrido-heterocycles The pyrido-heterocycles can be used for treating cancer (cervix, kidney, lung, breast and epidermal skin) and multi-drug resistant tuberculosis. These heterocycles can also be used as anti-biofilm agents against pathogenic strains, which will minimize the risk of secondary infections.

专利号:US-8697876-B2
优先权日:2010-04-02
标 题:Compositions and methods of synthesis of pyridinolypiperidine 5-HT1F agonists
发明人：CARNIAUX JEAN-FRANCOIS; CUMMINS JONATHAN
权利人:CARNIAUX JEAN-FRANCOIS; CUMMINS JONATHAN; COLUCID PHARMACEUTICALS INC
摘要:The present invention provides a novel polymorph of the hemisuccinate salt of 2,4,6-trifluoro-N-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide (Form A) characterized by a unique X-ray diffraction pattern and Differential Scanning Calorimetry profile, as well as a unique crystalline structure. This polymorph is useful in pharmaceutical compositions, for example, for the treatment and prevention of migraine. The invention also provides a process for the synthesis of pyridinoylpiperidine compounds of Formula I in high yield and high purity. In particular, the provides a process for the preparation of 2,4,6-trifluoro-N-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide, its hemisuccinate salt and polymorph (Form A).

专利号:US-2006211858-A1
优先权日:2001-02-28
标 题 :Novel substituted calix (4) pyrroles and process for the synthesis of calix (4) pyrroles over molecular sieve catalysts
发明人：RAGHAVAN KONDAPURAM V; KULKARNI SHIVANAND J; KISHAN MOTKURI R; SRINIVAS NAGABANDI
权利人:RAGHAVAN KONDAPURAM V; KULKARNI SHIVANAND J; KISHAN MOTKURI R; SRINIVAS NAGABANDI
摘要:The present invention relates to novel calix pyrroles and a process for synthesis of calix (4) pyrroles by reacting pyrrole with cyclic or acyclic ketones in dichloro methane (DCM) solvent over molecular sieve catalysts which provides an eco-friendly, more economical and selective heterogeneous method.

专利号:US-2006183758-A1
优先权日:2005-02-17
标 题:Method for synthesis of AZA-annelated pyrroles, thiophenes, and furans
发明人：BEARD CHARLES D; LEE VING J; WHITTLE C E
权利人:CB RES AND DEV INC
摘要:Methods of synthesis of intermediates that are useful as bioisosteres of the indole, benzofuran and benzothiophene scaffold are disclosed.

专利号:US-6605194-B2
优先权日:2001-02-26
标 题:Substituted calix (4) pyrroles and process for the synthesis of calix (4) pyrroles over molecular sieve catalysts
发明人：RAGHAVAN KONDAPURAM VIJAYA; KULKARNI SHIVANAND JANARDAN; KISHAN MOTKURI RADHA; SRINIVAS NAGABANDI
权利人:COUNCIL SCIENT IND RES
摘要:The present invention relates to novel calix pyrroles and a process for synthesis of calix (4) pyrroles by reacting pyrrole with cyclic or acyclic ketones in dichloro methane (DCM) solvent over molecular sieve catalysts which provides an eco-friendly, more economical and selective heterogeneous method.

专利号:WO-2022191172-A1
优先权日:2021-03-09
标题:Linker and carrier for nucleic acid solid phase synthesis
发明人：HARI YOSHIYUKI; FUCHI YASUFUMI; YAMAMOTO KAZUKI; ITO YUTA
权利人:LIID PHARMACEUTICALS INC
摘要:The present invention provides: a universal linker for synthesis of a nucleic acid solid phase, represented by formula (I), which makes it possible to suppress the occurrence of byproducts and which makes it possible to synthesize DNA and RNA of high purity with greater efficiency; and a carrier for nucleic acid solid phase synthesis which carries the linker. [In the formula, each symbol is as defined in the description.]